EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
3.4.16.2 | 0.0000003 |
- |
[4-[1-(3-chloro-4-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl][(1R,2R,4S)-2-(2,4-difluorophenyl)-4-(dimethylamino)-4-methylcyclopentyl]methanone |
pH not specified in the publication, temperature not specified in the publication |
731431 |
3.4.16.2 | 0.0000004 |
- |
[(3S,4R)-1-tert-butyl-4-(2,4-difluorophenyl)pyrrolidin-3-yl](4-[(1Z)-1-[(2,5-dichlorophenyl)amino]-3-iminobut-1-en-1-yl]piperidin-1-yl)methanone |
pH not specified in the publication, temperature not specified in the publication |
731430 |
3.4.16.2 | 0.0000005 |
- |
[(3S,4R)-1-tert-butyl-4-(2,4-difluorophenyl)pyrrolidin-3-yl](4-[(1Z)-1-[(3-chloro-4-fluorophenyl)amino]-3-iminoprop-1-en-1-yl]piperidin-1-yl)methanone |
pH not specified in the publication, temperature not specified in the publication |
731430 |
3.4.16.2 | 0.0000009 |
- |
[(3S,4R)-1-tert-butyl-4-(2,4-difluorophenyl)pyrrolidin-3-yl](4-[(1Z)-1-[(2,5-dichlorophenyl)amino]-3-iminobut-1-en-1-yl]piperidin-1-yl)methanone |
in 100% mouse plasma, pH not specified in the publication, temperature not specified in the publication |
731430 |
3.4.16.2 | 0.0000013 |
- |
[4-[1-(3-chloro-4-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl][(1R,2R,4S)-2-(2,4-difluorophenyl)-4-(dimethylamino)-4-methylcyclopentyl]methanone |
in 100% mouse plasma, pH not specified in the publication, temperature not specified in the publication |
731431 |
3.4.16.2 | 0.0000014 |
- |
[(3S,4R)-1-tert-butyl-4-(2,4-difluorophenyl)pyrrolidin-3-yl](4-[(1Z)-1-[(3-chloro-4-fluorophenyl)amino]-3-iminoprop-1-en-1-yl]piperidin-1-yl)methanone |
in 100% mouse plasma, pH not specified in the publication, temperature not specified in the publication |
731430 |
3.4.16.2 | 0.0037 |
- |
N-benzyloxycarbonyl-Pro-prolinal |
pH 5.6, 30°C |
731918 |