EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
3.4.14.1 | 0.0000002 |
- |
N-[(1E,3S)-5-phenyl-1-(phenylsulfonyl)pent-1-en-3-yl]-L-norvalinamide |
- |
707715 |
3.4.14.1 | 0.0000015 |
- |
(2S)-2-amino-N-[(1S)-2-(biphenyl-4-yl)-1-cyanoethyl]butanamide |
- |
707715 |
3.4.14.1 | 0.000045 |
- |
1-(2S-2-aminobutanoyl)-4-(2S-N-(2S-3-(m-fluorophenyl)propan-2-yl-amide)4-phenylbutan-2-yl-amide)semicarbazide |
- |
664305 |
3.4.14.1 | 0.0018 |
- |
N2-(morpholin-4-ylcarbonyl)-N-[(1E,3S)-5-phenyl-1-(phenylsulfonyl)pent-1-en-3-yl]-L-leucinamide |
- |
707715 |
3.4.14.1 | 0.0055 |
- |
3-chloro-2-hydroxypropyl (2Z)-2-(2-aminoacetamido)-3-phenylprop-2-enoate |
pH 5.0, 37°C |
754604 |
3.4.14.1 | 0.017 |
- |
prop-2-en-1-yl 2-(2-amino-3-phenylpropanamido)prop-2-enoate |
pH 5.0, 37°C |
754604 |
3.4.14.1 | 0.05 |
- |
Gly-DELTAZPhe-Gly-DELTAEPhe-Gly |
at 37°C in acetate buffer (pH 5) containing NaCl (10 mM) |
699734 |
3.4.14.1 | 0.122 |
- |
Gly-DELTAZPhe-Gly-DELTAEPhe-Phe |
at 37°C in acetate buffer (pH 5) containing NaCl (10 mM) |
699734 |
3.4.14.1 | 0.173 |
- |
Gly-DELTAZPhe-Gly-DELTAEPhe-Gly-OMe |
at 37°C in acetate buffer (pH 5) containing NaCl (10 mM) |
699734 |
3.4.14.1 | 0.324 |
- |
Gly-DELTAZPhe-Gly-DELTAEPhe-Phe-OMe |
at 37°C in acetate buffer (pH 5) containing NaCl (10 mM) |
699734 |