EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
2.8.2.2 | -999 |
- |
more |
inhibition kinetics |
761001 |
2.8.2.2 | -999 |
- |
more |
inhibition kinetics and modeling, detailed overview |
761727 |
2.8.2.2 | 0.0002 |
- |
bazedoxifene |
liver cytosol, pH 7.4, 37°C, substrate lithocholic acid, noncompetitive inhibition |
761727 |
2.8.2.2 | 0.0005 |
- |
raloxifene |
liver cytosol, pH 7.4, 37°C, substrate lithocholic acid, noncompetitive inhibition |
761727 |
2.8.2.2 | 0.0006 |
- |
4'-hydroxy-2,3',4,5'-tetrachlorobiphenyl |
at pH 7.0 and 37°C |
738032 |
2.8.2.2 | 0.0007 |
- |
4'-hydroxy-2,5-dichlorobiphenyl |
at pH 7.0 and 37°C |
738032 |
2.8.2.2 | 0.0007 |
- |
androsterone |
pH 7.0, 25°C, recombinant wild-type enzyme |
694259 |
2.8.2.2 | 0.0008 |
- |
4-hydroxy-2',3,5-trichlorobiphenyl |
at pH 7.0 and 37°C |
738032 |
2.8.2.2 | 0.0008 |
- |
arzoxifene |
liver cytosol, pH 7.4, 37°C, substrate lithocholic acid, mixed inhibition |
761727 |
2.8.2.2 | 0.0008 |
- |
lasofoxifene |
liver cytosol, pH 7.4, 37°C, substrate lithocholic acid, noncompetitive inhibition |
761727 |