EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
2.7.7.65 | 0.0005 |
- |
cyclic di-3',5'-guanylate |
wild-type |
682885 |
2.7.7.65 | 0.0009 |
- |
cyclic di-3',5'-guanylate |
mutant R313A |
682885 |
2.7.7.65 | 0.0028 |
- |
cyclic di-3',5'-guanylate |
mutant R148A, 30°C, pH 8.0 |
680703 |
2.7.7.65 | 0.0029 |
- |
cyclic di-3',5'-guanylate |
mutant R148A/R178A, 30°C, pH 8.0 |
680703 |
2.7.7.65 | 0.0036 |
- |
cyclic di-3',5'-guanylate |
mutant R178A, 30°C, pH 8.0 |
680703 |
2.7.7.65 | 0.005 |
- |
3-O-alpha-L-rhamnopyranosyl-(1-2)-beta-D-galactopyranosyl-(1-2)-beta-D-glucuronopyranosyl soyasapogenol B 22-O-alpha-D-glucopyranoside |
pH 7.5, 30°C |
682338 |
2.7.7.65 | 0.005 |
- |
cyclic di-3',5'-guanylate |
double mutant R148A/R178A |
682885 |
2.7.7.65 | 0.0058 |
- |
cyclic di-3',5'-guanylate |
wild-type, 30°C, pH 8.0 |
680703 |
2.7.7.65 | 0.033 |
- |
cyclic di-3',5'-guanylate |
triple mutant R148A/R178A/R313A |
682885 |
2.7.7.65 | 0.07 |
- |
papulacandin B |
pH 7.5, 30°C |
682338 |