EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
2.7.7.18 | -999 |
- |
more |
inhibition kinetics, overview |
738672 |
2.7.7.18 | 0.0079 |
- |
K891-0166 |
pH 7.5, 37°C |
727776 |
2.7.7.18 | 0.024 |
- |
2-(2,4-dimethylphenyl)-N-(4-([(5-methyl-3-isoxazolyl)amino]sulfonyl)phenyl)-4-quinolinecarboxamide |
pH 7.5, 37°C, recombinant mutant T12A |
738672 |
2.7.7.18 | 0.03 |
- |
2-(2,4-dimethylphenyl)-N-(4-([(5-methyl-3-isoxazolyl)amino]sulfonyl)phenyl)-4-quinolinecarboxamide |
pH 7.5, 37°C, recombinant mutant W117A |
738672 |
2.7.7.18 | 0.035 |
- |
2-(2,4-dimethylphenyl)-N-(4-([(5-methyl-3-isoxazolyl)amino]sulfonyl)phenyl)-4-quinolinecarboxamide |
pH 7.5, 37°C, recombinant wild-type enzyme |
738672 |
2.7.7.18 | 0.037 |
- |
2-(2,4-dimethylphenyl)-N-(4-([(5-methyl-3-isoxazolyl)amino]sulfonyl)phenyl)-4-quinolinecarboxamide |
pH 7.5, 37°C, recombinant mutant P44A |
738672 |
2.7.7.18 | 0.056 |
- |
2-(2,4-dimethylphenyl)-N-(4-([(5-methyl-3-isoxazolyl)amino]sulfonyl)phenyl)-4-quinolinecarboxamide |
pH 7.5, 37°C, recombinant mutant W45A |
738672 |
2.7.7.18 | 0.094 |
- |
2-(2,4-dimethylphenyl)-N-(4-([(5-methyl-3-isoxazolyl)amino]sulfonyl)phenyl)-4-quinolinecarboxamide |
pH 7.5, 37°C, recombinant mutant K47A |
738672 |
2.7.7.18 | 0.114 |
- |
2-(2,4-dimethylphenyl)-N-(4-([(5-methyl-3-isoxazolyl)amino]sulfonyl)phenyl)-4-quinolinecarboxamide |
pH 7.5, 37°C, recombinant mutant T86A |
738672 |