EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
2.7.4.2 | -999 |
- |
more |
inhibition kinetics, product inhibition patterns |
671609 |
2.7.4.2 | 0.0077 |
- |
phosphomevalonate |
pH 7.0, 25°C |
645183 |
2.7.4.2 | 0.014 |
- |
5-diphosphomevalonate |
pH 7.0, 25°C |
645183 |
2.7.4.2 | 0.018 |
- |
(R)-5-diphosphomevalonate |
wild-type, 30°C, pH 8.0 |
672221 |
2.7.4.2 | 0.018 |
- |
mevalonate 5-diphosphate |
pH 7.0, 30°C, recombinant wild-type enzyme |
672221 |
2.7.4.2 | 0.137 |
- |
ATP |
pH 7.0, 25°C |
645183 |
2.7.4.2 | 0.41 |
- |
ADP |
pH 7.0, 25°C |
645183 |
2.7.4.2 | 0.806 |
- |
(R)-5-diphosphomevalonate |
mutant R111M, 30°C, pH 8.0 |
672221 |
2.7.4.2 | 0.806 |
- |
mevalonate 5-diphosphate |
pH 7.0, 30°C, recombinant mutant R111M |
672221 |
2.7.4.2 | 1.14 |
- |
(R)-5-diphosphomevalonate |
mutant R84M, 30°C, pH 8.0 |
672221 |