EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
2.7.11.2 | -999 |
- |
more |
- |
642159 |
2.7.11.2 | -999 |
- |
more |
dichloroacetate inhibition kinetics and EC50 values with wild-type and mutant PDHK2s |
673688 |
2.7.11.2 | -999 |
- |
more |
inhibition kinetics |
661094 |
2.7.11.2 | -999 |
- |
more |
inhibition kinetics for thiamine diphosphate |
642143 |
2.7.11.2 | -999 |
- |
more |
isozyme PDK4: K+ reduces the Ki for ADP and therefor enhances the inhibitory affect |
642159 |
2.7.11.2 | -999 |
- |
more |
Ki value for ADP depends on the presence and concentration of monovalent cations, e.g. NH4+ or K+ |
642134 |
2.7.11.2 | 0.0031 |
- |
adenosine 5'-[beta,gamma-imido]triphosphate |
pH 7.4, 30°C, versus ATP |
661094 |
2.7.11.2 | 0.1 |
- |
ADP |
pH 7.5, 30°C |
642133 |
2.7.11.2 | 0.14 |
0.52 |
ADP |
pH 7.4, 30°C, versus ATP, dependent on the assay conditions concerning buffer composition, overview |
661094 |
2.7.11.2 | 0.2 |
- |
ADP |
37°C, recombinant isozyme PDK2 wild-type |
642153 |