EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
2.7.1.145 | -999 |
- |
more |
feedback inhibition kinetics |
661072 |
2.7.1.145 | -999 |
- |
more |
inhibition kinetics, overview |
662607 |
2.7.1.145 | 0.00066 |
- |
(E)-5-(2-bromovinyl)-2'-deoxyuridine |
pH 7.6, 30°C, reaction with thymidine, fusion protein with glutathione S-transferase |
636843 |
2.7.1.145 | 0.001 |
- |
2'-deoxycytidine |
pH 8.0, 22°C, competitive with thymidine |
636839, 636840 |
2.7.1.145 | 0.001 |
- |
thymidine |
pH 8.0, 22°C, competitive with 2'-deoxycytidine |
636839, 636840 |
2.7.1.145 | 0.002 |
- |
thymidine |
pH 8.0, 22°C, reaction with 2'-deoxyadenosine |
636840 |
2.7.1.145 | 0.003 |
- |
thymidine |
pH 8.0, 22°C, reaction with 2'-deoxyguanosine |
636840 |
2.7.1.145 | 0.0047 |
- |
dTTP |
uncompetitive versus 2'-deoxythymidine, recombinant wild-type enzyme |
661702 |
2.7.1.145 | 0.005 |
- |
TTP |
pH 8.0, 22°C |
636839 |
2.7.1.145 | 0.0163 |
- |
dTTP |
competitive versus ATP, recombinant wild-type enzyme |
661702 |