EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
2.4.2.4 | 0.000002 |
- |
5-chloro-6-[1-(2-iminopyrrolidinyl)methyl] uracil hydrochloride |
- |
658387 |
2.4.2.4 | 0.000011 |
- |
5-fluoro-6-[(2-aminoimidazol-1-yl)methyl]uracil |
- |
702614 |
2.4.2.4 | 0.000017 |
- |
5-fluoro-6-[(2-aminoimidazol-1-yl)methyl]uracil |
- |
702614 |
2.4.2.4 | 0.00002 |
- |
5-chloro-6-[1-(imminopyrrolidinyl)methyl]uracil hydrochloride |
- |
638468 |
2.4.2.4 | 0.00002 |
- |
thymidine phosphorylase inhibitor |
- |
658657 |
2.4.2.4 | 0.000051 |
- |
5-fluoro-6-(1H-imidazol-1-ylmethyl)pyrimidine-2,4(1H,3H)-dione |
- |
676235 |
2.4.2.4 | 0.000165 |
- |
6-(2-aminoethyl)amine-5-chlorouracil |
- |
638467 |
2.4.2.4 | 0.000236 |
- |
(4xi)-5-methyl-2',3'-O-[(1R)-2-phosphonoethylidene]cytidine |
- |
675314 |
2.4.2.4 | 0.00037 |
- |
5-fluoro-6-[(4H-1,2,4-triazol-4-ylamino)methyl]pyrimidine-2,4(1H,3H)-dione |
- |
676235 |
2.4.2.4 | 0.00077 |
- |
[(2S,3aR,4R,6R,6aR)-4-(5-chloro-2,4-dioxo-3,4-dihydropyrimidin-1(2H)-yl)-6-(hydroxymethyl)tetrahydrofuro[3,4-d][1,3]dioxol-2-yl]phosphonic acid |
- |
689263 |