EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
2.4.2.4 | -999 |
- |
more |
inhibition kinetics |
759338 |
2.4.2.4 | -999 |
- |
more |
inhibition kinetics, Lineweaver-Burk plots |
758893, 760047 |
2.4.2.4 | -999 |
- |
more |
inhibition kinetics, overview |
702614 |
2.4.2.4 | 0.0000013 |
- |
5-chloro-6-(2-iminopyrrolidin-1-yl)methyl-2,4-(1H,3H)-pyrimidine |
enzyme purified from V79 cells, in 20 mM Bis-Tris-HCl (pH 6.4), at 37°C |
688264 |
2.4.2.4 | 0.000002 |
- |
5-chloro-6-[1-(2-iminopyrrolidinyl)methyl] uracil hydrochloride |
- |
658387 |
2.4.2.4 | 0.0000021 |
- |
5-chloro-6-(2-iminopyrrolidin-1-yl)methyl-2,4-(1H,3H)-pyrimidine |
enzyme purified from placenta, in 20 mM Bis-Tris-HCl (pH 6.4), at 37°C |
688264 |
2.4.2.4 | 0.000011 |
- |
5-fluoro-6-[(2-aminoimidazol-1-yl)methyl]uracil |
- |
702614 |
2.4.2.4 | 0.000017 |
- |
5-fluoro-6-[(2-aminoimidazol-1-yl)methyl]uracil |
- |
702614 |
2.4.2.4 | 0.00002 |
- |
5-chloro-6-[1-(2-iminopyrrolidinyl)methyl] uracil hydrochloride |
pH and temperature not specified in the publication |
759610 |
2.4.2.4 | 0.00002 |
- |
5-chloro-6-[1-(imminopyrrolidinyl)methyl]uracil hydrochloride |
- |
638468 |