EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
2.4.2.26 | -999 |
- |
more |
competitive inhibition of the acceptor substrates |
637614 |
2.4.2.26 | 0.00007 |
- |
heparin |
pH 6.5, 37°C, mutant enzyme D745E |
659394 |
2.4.2.26 | 0.00011 |
- |
heparin |
pH 6.5, 37°C, mutant enzyme D747E |
659394 |
2.4.2.26 | 0.00011 |
- |
heparin |
pH 6.5, 37°C, mutant enzyme W746N |
659394 |
2.4.2.26 | 0.00012 |
- |
heparin |
pH 6.5, 37°C, mutant enzyme W746G |
659394 |
2.4.2.26 | 0.00012 |
- |
heparin |
pH 6.5, 37°C, wild-type enzyme |
659394 |
2.4.2.26 | 0.00013 |
- |
heparin |
pH 6.5, 37°C, mutant enzyme W746D |
659394 |
2.4.2.26 | 0.00014 |
- |
heparin |
pH 6.5, 37°C, mutant enzyme D316G |
659394 |
2.4.2.26 | 0.00015 |
- |
heparin |
pH 6.5, 37°C, mutant enzyme D314G |
659394 |
2.4.2.26 | 0.00015 |
- |
heparin |
pH 6.5, 37°C, mutant enzyme D747G |
659394 |