EC Number   |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
|---|
    2.4.2.17 | 0.0005 |
- |
L-histidine |
wild type enzyme, at pH 8.5 and 30°C |
736541 |
| 2.4.2.17 | 0.002 |
- |
1-[(5,6-diphenyl-1,2,4-triazin-3-yl)sulfanyl]-3-(1,3-thiazol-2-yl)propan-2-one |
- |
705015 |
| 2.4.2.17 | 0.002 |
- |
N-[3-[(6-nitro-1,3-benzothiazol-2-yl)amino]-3-oxo-1-phenylpropyl]benzamide |
- |
705015 |
| 2.4.2.17 | 0.004 |
- |
L-histidine |
uncompetitive versus ATP, pH 8.0, 25°C |
721673 |
| 2.4.2.17 | 0.0079 |
- |
L-histidine |
uncompetitive versus ATP, pH 8.25, 25°C |
721673 |
| 2.4.2.17 | 0.011 |
- |
L-histidine |
mutant enzyme A270D, at pH 8.5 and 30°C |
736541 |
| 2.4.2.17 | 0.022 |
- |
L-histidine |
mutant enzyme S232Y, at pH 8.5 and 30°C |
736541 |
| 2.4.2.17 | 0.0235 |
- |
L-histidine |
Kii-value, non competitive versus 5-phospho-alpha-D-ribosyl diphosphate, pH 8.5, 25°C |
721673 |
| 2.4.2.17 | 0.0257 |
- |
L-histidine |
Kis-value, non competitive versus 5-phospho-alpha-D-ribosyl diphosphate, pH 8.5, 25°C |
721673 |
| 2.4.2.17 | 0.0269 |
- |
L-histidine |
uncompetitive versus ATP, pH 8.75, 25°C |
721673 |
