EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
1.13.12.13 | 0.022 |
- |
coelenterazine |
pH and temperature not specified in the publication |
764497 |
1.13.12.13 | 0.035 |
- |
8-benzyl-6-(3-hydroxyphenyl)-2-[(4-hydroxyphenyl)methyl]imidazo[1,2-a]pyrazin-3(7H)-one |
pH and temperature not specified in the publication |
764497 |
1.13.12.13 | 0.04 |
- |
2-[(5-methylfuran-2-yl)methyl]-8-[(3-fluorophenyl)methyl]-6-phenylimidazo[1,2-a]pyrazin-3(7H)-one |
pH and temperature not specified in the publication |
764497 |
1.13.12.13 | 0.058 |
- |
8-benzyl-2-[(2-fluorophenyl)methyl]-6-phenylimidazo[1,2-a]pyrazin-3(7H)-one |
pH and temperature not specified in the publication |
764497 |
1.13.12.13 | 0.06 |
- |
2-[(5-ethylfuran-2-yl)methyl]-8-[(3-fluorophenyl)methyl]-6-phenylimidazo[1,2-a]pyrazin-3(7H)-one |
pH and temperature not specified in the publication |
764497 |
1.13.12.13 | 0.06 |
- |
8-[(2-fluorophenyl)methyl]-2-[(5-methylfuran-2-yl)methyl]-6-phenylimidazo[1,2-a]pyrazin-3(7H)-one |
pH and temperature not specified in the publication |
764497 |
1.13.12.13 | 0.063 |
- |
6-(2-fluorophenyl)-8-[(4-fluorophenyl)methyl]-2-[(5-methylfuran-2-yl)methyl]imidazo[1,2-a]pyrazin-3(7H)-one |
pH and temperature not specified in the publication |
764497 |
1.13.12.13 | 0.064 |
- |
8-[(3,5-difluorophenyl)methyl]-2-[(5-methylfuran-2-yl)methyl]-6-phenylimidazo[1,2-a]pyrazin-3(7H)-one |
pH and temperature not specified in the publication |
764497 |
1.13.12.13 | 0.08 |
- |
8-[(2,3-difluorophenyl)methyl]-2-[(5-methylfuran-2-yl)methyl]-6-phenylimidazo[1,2-a]pyrazin-3(7H)-one |
pH and temperature not specified in the publication |
764497 |
1.13.12.13 | 0.084 |
- |
8-benzyl-2-[(furan-2-yl)methyl]-6-(3-hydroxyphenyl)imidazo[1,2-a]pyrazin-3(7H)-one |
pH and temperature not specified in the publication |
764497 |