EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
1.1.1.213 | -999 |
- |
more |
more Ki values given for different inhibitors of androsterone oxidation, 9,10-phenanthrenequinone- and 5alpha-androstane-3,17-dione reduction |
347982 |
1.1.1.213 | 0.00001 |
- |
Cibacron blue |
slope effect, 0.025 mM androsterone, varying NADP+ concentrations |
286355 |
1.1.1.213 | 0.000107 |
- |
2-(2,4-dioxo-1,3-thiazolidin-5-yl)-N-(2-hydroxyphenyl)acetamide |
pH 7.0, temperature not specified in the publication |
725671 |
1.1.1.213 | 0.0002 |
- |
Cibacron blue |
slope effect, 0.25 mM NADP+, varying androsterone concentrations |
286355 |
1.1.1.213 | 0.0002 |
- |
indomethacin |
competitive, for 9,10-phenanthrenequinone and 5alpha-androstane-3,17-dione reduction at pH 6.0 |
347982 |
1.1.1.213 | 0.0005 |
- |
Cibacron blue |
intercept effect, 0.25 mM NADP+, varying androsterone concentrations |
286355 |
1.1.1.213 | 0.00057 |
- |
indomethacin |
- |
347979 |
1.1.1.213 | 0.0008 |
- |
Prostaglandin B1 |
androsterone oxidation |
347982 |
1.1.1.213 | 0.000835 |
- |
indomethacin |
competitive for androstene oxidation at pH 7.0. IC50 is 0.003 mM at H 7.0, 0.045 at pH 9.0 |
347982 |
1.1.1.213 | 0.001 |
- |
indomethacin |
- |
347980 |