EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
1.1.1.141 | -999 |
- |
more |
0.0189, endogenous mixture of palmitic, stearic, oleic and linoleic acid |
285933 |
1.1.1.141 | -999 |
- |
more |
inhibition kinetics |
285916 |
1.1.1.141 | 0.00009 |
- |
5-[4-(cyclohexylethoxy)benzylidene]-2,4-thiazolidenedione |
37°C, pH 7.5 |
654348 |
1.1.1.141 | 0.00011 |
- |
5-[4-(cyclohexylpropoxy)benzylidene]-2,4-thiazolidenedione |
37°C, pH 7.5 |
654348 |
1.1.1.141 | 0.00027 |
- |
5-[4-(cyclohexylmethoxy)benzylidene]-2,4-thiazolidenedione |
37°C, pH 7.5 |
654348 |
1.1.1.141 | 0.0006 |
- |
5-[4-((1-methyl)-cyclohexylmethoxy)benzylidene]-2,4-thiazolidenedione |
37°C, pH 7.5 |
654348 |
1.1.1.141 | 0.0009 |
- |
5-[4-(cyclohexyloxy)benzylidene]-2,4-thiazolidenedione |
37°C, pH 7.5 |
654348 |
1.1.1.141 | 0.0012 |
- |
5-[4-(benzoxy)benzylidene]-2,4-thiazolidenedione |
37°C, pH 7.5 |
654348 |
1.1.1.141 | 0.0022 |
- |
5-[4-((1-methyl)-cyclohexylmethoxy)benzyl]-2,4-thiazolidenedione |
37°C, pH 7.5 |
654348 |
1.1.1.141 | 0.005 |
- |
5-[4-(cyclohexylbutoxy)benzylidene]-2,4-thiazolidenedione |
37°C, pH 7.5 |
654348 |