EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
3.6.1.12 | 0.356 |
- |
5-hydroxytriptonide |
in 50 mM Tris, pH 8.0, 100 mM KCl, 5 mM MgCl2, 100 mg/ml bovine serum albumin, 1 mM dithiothreitol, at 37°C |
719287 |
3.6.1.12 | -999 |
- |
more |
inhibition kinetics |
755792 |
3.6.1.12 | 0.168 |
- |
triptolide |
in 50 mM Tris, pH 8.0, 100 mM KCl, 5 mM MgCl2, 100 mg/ml bovine serum albumin, 1 mM dithiothreitol, at 37°C |
719287 |
3.6.1.12 | 0.135 |
- |
triptonide |
in 50 mM Tris, pH 8.0, 100 mM KCl, 5 mM MgCl2, 100 mg/ml bovine serum albumin, 1 mM dithiothreitol, at 37°C |
719287 |
3.6.1.12 | 0.085 |
- |
triptriolide |
in 50 mM Tris, pH 8.0, 100 mM KCl, 5 mM MgCl2, 100 mg/ml bovine serum albumin, 1 mM dithiothreitol, at 37°C |
719287 |