EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
3.4.24.82 | 0.000105 |
- |
GGWGPWGPWGDCSRTCGGG |
- |
638958 |
3.4.24.82 | 0.0000033 |
- |
tissue inhibitor of matrix metalloproteinases-3 |
- |
668343 |
3.4.24.82 | 0.00002 |
- |
tinzaparin |
- |
668343 |
3.4.24.82 | 0.00008 |
- |
enoxaparin |
- |
668343 |
3.4.24.82 | 0.0000228 |
- |
SC81956 |
at 37°C |
678287 |
3.4.24.82 | 0.026 |
- |
QEYKAHHSYKLMS |
at 37°C |
678287 |
3.4.24.82 | 0.0000079 |
- |
TIMP-3 |
- |
680792 |
3.4.24.82 | -999 |
- |
more |
Ki(app) of N-terminal alanine-extension mutants and of position [-1] mutants of N-terminal inhibitory domain of tissue inhibitor of metalloproteinases 3 |
707445 |
3.4.24.82 | 0.00268 |
- |
(E)-4-[2-(3,5-dihydroxyphenyl)ethenyl]1,2-benzenediol |
pH 7.5, 37°C, substrate: C6-(Gly-Pro-Hyp-Pro-Hyp-Gly)2-Gly-Pro-Hyp-Gly-Thr-Lys(7-methoxycoumarin-4-yl)-Gly-GluLeuGluGly-ArgGly-Thr-Lys(Dnp)-Gly-Ile-Ser-(Gly-Pro-Hyp-Pro-Hyp-Gly)2-Gly-Pro-Hyp-NH2 |
708082 |
3.4.24.82 | 0.00506 |
- |
(E)-4-[2-(3,5-dihydroxyphenyl)ethenyl]1,2-benzenediol |
pH 7.5, 37°C, substrate: pH 7.5, 37°C, substrate: Lys(7-methoxycoumarin-4-yl)-Lys-Gln-Glu-Phe-Arg-Gly-Gln-Thr-Lys(Dnp)-NH2 |
708082 |