EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
3.4.24.82 | 0.000065 |
- |
(2R)-N4-hydroxy-2-(3-hydroxybenzyl)-N1-[(1S,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]butanediamide |
or above, pH not specified in the publication, temperature not specified in the publication |
734700 |
3.4.24.82 | 0.000003 |
- |
(2S,3R)-2-[(cyclopropylmethyl)amino]-N1-hydroxy-N4-[(1S,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]-3-methylbutanediamide |
or above, pH not specified in the publication, temperature not specified in the publication |
734700 |
3.4.24.82 | 0.00268 |
- |
(E)-4-[2-(3,5-dihydroxyphenyl)ethenyl]1,2-benzenediol |
pH 7.5, 37°C, substrate: C6-(Gly-Pro-Hyp-Pro-Hyp-Gly)2-Gly-Pro-Hyp-Gly-Thr-Lys(7-methoxycoumarin-4-yl)-Gly-GluLeuGluGly-ArgGly-Thr-Lys(Dnp)-Gly-Ile-Ser-(Gly-Pro-Hyp-Pro-Hyp-Gly)2-Gly-Pro-Hyp-NH2 |
708082 |
3.4.24.82 | 0.00506 |
- |
(E)-4-[2-(3,5-dihydroxyphenyl)ethenyl]1,2-benzenediol |
pH 7.5, 37°C, substrate: pH 7.5, 37°C, substrate: Lys(7-methoxycoumarin-4-yl)-Lys-Gln-Glu-Phe-Arg-Gly-Gln-Thr-Lys(Dnp)-NH2 |
708082 |
3.4.24.82 | 0.0453 |
- |
doxycycline |
rhADAMTS4(F213-R695), pH and temperature not specified in the publication |
709662 |
3.4.24.82 | 0.0611 |
- |
doxycycline |
rhADAMTS4(F213-A579), pH and temperature not specified in the publication |
709662 |
3.4.24.82 | 0.00008 |
- |
enoxaparin |
- |
668343 |
3.4.24.82 | 0.000105 |
- |
GGWGPWGPWGDCSRTCGGG |
- |
638958 |
3.4.24.82 | 0.000079 |
- |
marimastat |
pH not specified in the publication, temperature not specified in the publication |
734700 |
3.4.24.82 | 0.0869 |
- |
minocycline |
rhADAMTS4(F213-R695), pH and temperature not specified in the publication |
709662 |