EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
3.4.23.20 | 0.11 |
- |
methyl (2S)-2-({hydroxy[({N-[(naphthalen-1-yl)acetyl]-L-valyl}amino)methyl]phosphoryl}oxy)-3-phenylpropanoate |
- |
649272 |
3.4.23.20 | 0.0008 |
- |
methyl (2S)-2-({[(4S,7R)-2,5-dioxo-4-(propan-2-yl)-2,3,4,5,6,7-hexahydro-1H-8,10-etheno-3,6-benzodiazacycloundecin-7-yl](hydroxy)phosphoryl}oxy)-3-phenylpropanoate |
- |
649272 |
3.4.23.20 | 0.0076 |
- |
methyl (2S)-2-({[(R)-[(N-formyl-L-valyl)amino](naphthalen-2-yl)methyl](hydroxy)phosphoryl}oxy)-3-phenylpropanoate |
- |
649272 |
3.4.23.20 | 0.0000001 |
- |
methyl cyclo[(2S)-2-[[(1R)-1-(N-(l-N-(3-methylbutanoyl)valyl-L-aspartyl)amino)-3-methylbutyl]ydroxyphosphinyloxy]-3-(3-aminomethyl)] phenylpropanoate |
pH 4.6, macrocyclic pentapeptide inhibitor |
649841 |
3.4.23.20 | 0.00000001 |
- |
pepstatin |
pH 5.0, 37°C, wild-type Pencillopepsin JT-2 |
653829 |
3.4.23.20 | 0.0000004 |
- |
pepstatin |
pH 5.0, 37°C, mutant T219S |
653829 |
3.4.23.20 | 0.00055 |
- |
pepstatin |
pH 5.0, 37°C, mutant T219A |
653829 |
3.4.23.20 | 0.0016 |
- |
pepstatin |
pH 5.0, 37°C, mutant T219V |
653829 |
3.4.23.20 | 0.0018 |
- |
pepstatin |
pH 5.0, 37°C, mutant T219G |
653829 |