EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
3.4.22.53 | 0.0898 |
- |
Ac-Thr-Pro-Leu-alpha-azaglycine-Ser-Pro-Pro-NH2 |
in 10 mM HEPES, 150 mM NaCl, 1 mM EDTA, pH 7.5, at 22°C |
732375 |
3.4.22.53 | 0.0087 |
- |
Ac-Thr-Pro-Leu-alpha-azaglycine-Ser-Pro-Pro-Pro-Ser-NH2 |
in 10 mM HEPES, 150 mM NaCl, 1 mM EDTA, pH 7.5, at 22°C |
732375 |
3.4.22.53 | 0.0072 |
- |
Ac-Thr-Pro-Leu-alpha-azaglycine-Ser-Pro-Pro-Pro-Ser-Pro-Arg-NH2 |
in 10 mM HEPES, 150 mM NaCl, 1 mM EDTA, pH 7.5, at 22°C |
732375 |
3.4.22.53 | 0.0035 |
- |
Ac-Thr-Ser-Leu-alpha-azaglycine-Ser-Pro-Pro-Pro-Ser-NH2 |
in 10 mM HEPES, 150 mM NaCl, 1 mM EDTA, pH 7.5, at 22°C |
732375 |
3.4.22.53 | 0.0058 |
- |
Ac-Thr-Trp-Leu-alpha-azaglycine-Ser-Pro-Pro-Pro-Ser-NH2 |
in 10 mM HEPES, 150 mM NaCl, 1 mM EDTA, pH 7.5, at 22°C |
732375 |
3.4.22.53 | 0.00206 |
- |
antipain |
room temperature, pH 7.5, with succinyl-Met-Leu-methylcoumarin as substrate |
644046 |
3.4.22.53 | 0.000286 |
- |
Cbz-Leu-DL-Abu-CONH-(CH2)3-(4-methylpiperazin-1-yl) |
in 50 mM Tris-HCl, 50 mM NaCl, 1 mM EDTA, 1 mM EGTA, 0.1% CHAPS, pH 7.5, 10 mM dithiothreitol, 5 mM CaCl2, and less than 5% (v/v) DMSO, temperature not specified in the publication |
717969 |
3.4.22.53 | 0.000077 |
- |
Cbz-Leu-DL-Abu-CONH-(CH2)3-2-methoxyadenin-9-yl |
in 50 mM Tris-HCl, 50 mM NaCl, 1 mM EDTA, 1 mM EGTA, 0.1% CHAPS, pH 7.5, 10 mM dithiothreitol, 5 mM CaCl2, and less than 5% (v/v) DMSO, temperature not specified in the publication |
717969 |
3.4.22.53 | 0.00007 |
- |
Cbz-Leu-DL-Abu-CONH-(CH2)3-adenin-9-yl |
in 50 mM Tris-HCl, 50 mM NaCl, 1 mM EDTA, 1 mM EGTA, 0.1% CHAPS, pH 7.5, 10 mM dithiothreitol, 5 mM CaCl2, and less than 5% (v/v) DMSO, temperature not specified in the publication |
717969 |
3.4.22.53 | 0.00114 |
- |
Cbz-Leu-DL-Abu-CONH-(CH2)3-cytosin-3-yl |
in 50 mM Tris-HCl, 50 mM NaCl, 1 mM EDTA, 1 mM EGTA, 0.1% CHAPS, pH 7.5, 10 mM dithiothreitol, 5 mM CaCl2, and less than 5% (v/v) DMSO, temperature not specified in the publication |
717969 |