EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
4.2.1.10 | 0.000048 |
- |
(1R,4R,5R)-1,4,5-trihydroxy-3-[1-(2-hydroxyphenyl)-1H-1,2,3-triazol-4-yl]cyclohex-2-ene-1-carboxylic acid |
pH 7.5, 25°C |
716099 |
4.2.1.10 | 0.000054 |
- |
(1R,4R,5R)-1,4,5-trihydroxy-3-(3-nitrophenyl)cyclohex-2-ene-1-carboxylic acid |
pH not specified in the publication, temperature not specified in the publication |
714752 |
4.2.1.10 | 0.000056 |
- |
(1R,2S,4S,5R)-2-(1-benzothiophen-5-yl)-1,4,5-trihydroxy-3-oxocyclohexanecarboxylic acid |
pH 7.0, 25°C, 50 mM Tris-HOAc |
703225 |
4.2.1.10 | 0.000073 |
- |
(1R,4R,5R)-1,4,5-trihydroxy-3-[1-(thiophen-2-ylmethyl)-1H-1,2,3-triazol-4-yl]cyclohex-2-ene-1-carboxylic acid |
pH 7.5, 25°C |
716099 |
4.2.1.10 | 0.000074 |
- |
(1R,2S,4S,5R)-2-[difluoro(pentafluorophenyl)methyl]-1,4,5-trihydroxy-3-oxocyclohexanecarboxylic acid |
pH 7.0, 25°C, 50 mM Tris-HOAc |
703225 |
4.2.1.10 | 0.000078 |
- |
(1R,4R,5R)-1,4,5-trihydroxy-3-[1-(3-nitrophenyl)-1H-1,2,3-triazol-4-yl]cyclohex-2-ene-1-carboxylic acid |
pH 7.5, 25°C |
716099 |
4.2.1.10 | 0.000089 |
- |
(1R,2R,4S,5R)-1,4,5-trihydroxy-2-(4-methylbenzyl)-3-oxocyclohexanecarboxylic acid |
pH 7.0, 25°C, 50 mM Tris-HOAc |
703225 |
4.2.1.10 | 0.00009 |
- |
(1R,2S,4S,5R)-1,4,5-trihydroxy-2-(4-methylbenzyl)-3-oxocyclohexanecarboxylic acid |
pH 7.0, 25°C, 50 mM Tris-HOAc |
703225 |
4.2.1.10 | 0.00009 |
- |
(1R,2S,4S,5R)-2-benzyl-1,4,5-trihydroxy-3-oxocyclohexanecarboxylic acid |
pH 7.0, 25°C, 50 mM Tris-HOAc |
703225 |
4.2.1.10 | 0.0001 |
- |
(1R,2R,4S,5R)-2-benzyl-1,4,5-trihydroxy-3-oxocyclohexanecarboxylic acid |
pH 7.0, 25°C, 50 mM Tris·HCl |
703225 |