EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
3.4.24.82 | 0.00634 |
- |
pyrogallol |
pH 7.5, 37°C, substrate: C6-(Gly-Pro-Hyp-Pro-Hyp-Gly)2-Gly-Pro-Hyp-Gly-Thr-Lys(7-methoxycoumarin-4-yl)-Gly-GluLeuGluGly-ArgGly-Thr-Lys(Dnp)-Gly-Ile-Ser-(Gly-Pro-Hyp-Pro-Hyp-Gly)2-Gly-Pro-Hyp-NH2 |
708082 |
3.4.24.82 | 0.026 |
- |
QEYKAHHSYKLMS |
at 37°C |
678287 |
3.4.24.82 | 0.041 |
- |
pyrogallol |
pH 7.5, 37°C, substrate: Lys(7-methoxycoumarin-4-yl)-Lys-Gln-Glu-Phe-Arg-Gly-Gln-Thr-Lys(Dnp)-NH2 |
708082 |
3.4.24.82 | 0.0453 |
- |
doxycycline |
rhADAMTS4(F213-R695), pH and temperature not specified in the publication |
709662 |
3.4.24.82 | 0.0611 |
- |
doxycycline |
rhADAMTS4(F213-A579), pH and temperature not specified in the publication |
709662 |
3.4.24.82 | 0.0869 |
- |
minocycline |
rhADAMTS4(F213-R695), pH and temperature not specified in the publication |
709662 |
3.4.24.82 | 0.0973 |
- |
minocycline |
rhADAMTS4(F213-A579), pH and temperature not specified in the publication |
709662 |
3.4.24.82 | 0.12 |
- |
tetracycline |
rhADAMTS4(F213-A579), pH and temperature not specified in the publication |
709662 |
3.4.24.82 | 0.761 |
- |
tetracycline |
rhADAMTS4(F213-R695), pH and temperature not specified in the publication |
709662 |