EC Number   |
Ki Value [mM] |
Ki Value maximum [mM]  |
Inhibitor |
Reference |
|---|
   3.4.22.43 | 0.0011 |
- |
glycocitrine-IV |
in 100 mM sodium acetate buffer (pH 5.5) containing 5 mM EDTA and 5 mM dithioerythritol, at 27°C |
717374 |
| 3.4.22.43 | 0.0012 |
- |
1,3,5-trihydroxy-2,8-bis(3-methylbut-2-enyl)-10-methyl-9-acridone |
in 100 mM sodium acetate buffer (pH 5.5) containing 5 mM EDTA and 5 mM dithioerythritol, at 27°C |
717374 |
| 3.4.22.43 | 0.0017 |
- |
3,4-dihydro-3,5,8-trihydroxy-6-methoxy-2,2,7-trimethyl-2H-pyrano[2,3-a]acridin-12(7H)-one |
in 100 mM sodium acetate buffer (pH 5.5) containing 5 mM EDTA and 5 mM dithioerythritol, at 27°C |
717374 |
| 3.4.22.43 | 0.0042 |
- |
citrusinine-II |
in 100 mM sodium acetate buffer (pH 5.5) containing 5 mM EDTA and 5 mM dithioerythritol, at 27°C |
717374 |
| 3.4.22.43 | 0.0044 |
- |
2,3-dihydro-4,9-dihydroxy-2-(2-hydroxy-propan-2-yl)-11-methoxy-10-methylfuro[3,2-b]acridin-5(10H)-one |
in 100 mM sodium acetate buffer (pH 5.5) containing 5 mM EDTA and 5 mM dithioerythritol, at 27°C |
717374 |
| 3.4.22.43 | 0.01 |
- |
glycocitrine-I |
in 100 mM sodium acetate buffer (pH 5.5) containing 5 mM EDTA and 5 mM dithioerythritol, at 27°C |
717374 |
| 3.4.22.43 | 0.0102 |
- |
cathepsin V propeptide |
varying concentrations tested |
683207 |
