EC Number |
kcat/KM Value [1/mMs-1] |
kcat/KM Value Maximum [1/mMs-1] |
Substrate |
Reference |
---|
3.4.22.53 | 0.0394 |
- |
succinyl-Leu-Tyr-7-amido-4-methylcoumarin |
endoplasmic reticulum membrane m-calpain, in 100 mM imidazole-HCl buffer (pH 7.5), 5 mM L-cysteine, 2.5 mM 2-mercaptoethanol, 5 mM CaCl2, and 4% (v/v) dimethyl sulfoxide, at 30°C |
708960 |
3.4.22.53 | 0.0395 |
- |
succinyl-Leu-Tyr-7-amido-4-methylcoumarin |
endoplasmic reticulum lumen m-calpain, in 100 mM imidazole-HCl buffer (pH 7.5), 5 mM L-cysteine, 2.5 mM 2-mercaptoethanol, 5 mM CaCl2, and 4% (v/v) dimethyl sulfoxide, at 30°C |
708960 |
3.4.22.53 | 0.0399 |
- |
succinyl-Leu-Met-7-amido-4-methylcoumarin |
endoplasmic reticulum membrane m-calpain, in 100 mM imidazole-HCl buffer (pH 7.5), 5 mM L-cysteine, 2.5 mM 2-mercaptoethanol, 5 mM CaCl2, and 4% (v/v) dimethyl sulfoxide, at 30°C |
708960 |
3.4.22.53 | 0.0404 |
- |
succinyl-Leu-Met-7-amido-4-methylcoumarin |
endoplasmic reticulum lumen m-calpain, in 100 mM imidazole-HCl buffer (pH 7.5), 5 mM L-cysteine, 2.5 mM 2-mercaptoethanol, 5 mM CaCl2, and 4% (v/v) dimethyl sulfoxide, at 30°C |
708960 |
3.4.22.53 | 0.131 |
- |
t-butyloxycarbonyl-Val-Leu-Lys-7-amido-4-methylcoumarin |
endoplasmic reticulum membrane m-calpain, in 100 mM imidazole-HCl buffer (pH 7.5), 5 mM L-cysteine, 2.5 mM 2-mercaptoethanol, 5 mM CaCl2, and 4% (v/v) dimethyl sulfoxide, at 30°C |
708960 |
3.4.22.53 | 0.133 |
- |
t-butyloxycarbonyl-Val-Leu-Lys-7-amido-4-methylcoumarin |
endoplasmic reticulum lumen m-calpain, in 100 mM imidazole-HCl buffer (pH 7.5), 5 mM L-cysteine, 2.5 mM 2-mercaptoethanol, 5 mM CaCl2, and 4% (v/v) dimethyl sulfoxide, at 30°C |
708960 |
3.4.22.53 | 0.135 |
- |
succinyl-Leu-Leu-Val-Tyr-7-amido-4-methylcoumarin |
endoplasmic reticulum lumen m-calpain, in 100 mM imidazole-HCl buffer (pH 7.5), 5 mM L-cysteine, 2.5 mM 2-mercaptoethanol, 5 mM CaCl2, and 4% (v/v) dimethyl sulfoxide, at 30°C |
708960 |
3.4.22.53 | 0.137 |
- |
succinyl-Leu-Leu-Val-Tyr-7-amido-4-methylcoumarin |
endoplasmic reticulum membrane m-calpain, in 100 mM imidazole-HCl buffer (pH 7.5), 5 mM L-cysteine, 2.5 mM 2-mercaptoethanol, 5 mM CaCl2, and 4% (v/v) dimethyl sulfoxide, at 30°C |
708960 |