EC Number |
KM Value [mM] |
KM Value Maximum [mM] |
Substrate |
Reference |
---|
3.4.24.82 | 0.015 |
- |
5-carboxyfluorescein-Ala-Glu-Leu-Gln-Gly-Arg-Pro-Ile-Ser-Ile-Ala-Lys-N,N,N',N'-tetramethyl-6-carboxyrhodamine |
at pH 7.5 and 37°C |
754633 |
3.4.24.82 | 0.0203 |
- |
Aggrecan |
in 100 mM NaCl |
680792 |
3.4.24.82 | 0.0282 |
- |
chondroitin 4-sulfate |
in 100 mM NaCl |
680792 |
3.4.24.82 | 0.035 |
- |
Lys(carboxyfluorescein)-Asp-Val-Gln-Glu-Phe-Arg-Gly-Val-Thr-Ala-Val-Ile-Arg-Lys(tetramethylrhodamine)-Lys-Gly-Lys-NH2 |
pH 7.5, 37°C |
708082 |
3.4.24.82 | 0.0471 |
- |
[C6-(Gly-Pro-Hyp)5-Gly-Thr-Lys(7-amido-4-methylcoumarin)-Gly-Glu-Leu-Glu-Gly-Arg-Gly-Thr-Lys(2,4-dinitrophenyl)-Gly-Ile-Ser-(Gly-Pro-Hyp)5-NH2]3 |
ADAMTS-4-2, at 25°C |
680769 |
3.4.24.82 | 0.279 |
- |
C6-(Gly-Pro-Hyp-Pro-Hyp-Gly)2-Gly-Pro-Hyp-Gly-Thr-Lys(Mca)-Gly-Glu-Leu-Glu-Gly-Arg-Gly-Thr-Lys(Dnp)-Gly-Ile-Ser-(Gly-Pro-Hyp-Pro-Hyp-Gly)2-Gly-Pro-Hyp-NH2 |
ADAMTS-4-2, at 25°C |
680769 |
3.4.24.82 | 0.48 |
- |
QTVTWPDMELPLPRNITEGEARGSVILTVKPIFEVSPSPLK |
biotinylated peptide containing aggrecanase cleavage site |
638966 |
3.4.24.82 | 0.65 |
- |
[C6-(Gly-Pro-Hyp)5-Gly-Thr-Lys(7-amido-4-methylcoumarin)-Gly-Glu-Leu-Glu-Gly-Arg-Gly-Thr-Lys(2,4-dinitrophenyl)-Gly-Ile-Ser-(Gly-Pro-Hyp)5-NH2]3 |
ADAMTS-4-2, at 25°C |
680769 |
3.4.24.82 | 0.761 |
- |
C6-(Gly-Pro-Hyp-Pro-Hyp-Gly)2-Gly-Pro-Hyp-Gly-Thr-Lys(Mca)-Gly-Glu-Leu-Glu-Gly-Arg-Gly-Thr-Lys(Dnp)-Gly-Ile-Ser-(Gly-Pro-Hyp-Pro-Hyp-Gly)2-Gly-Pro-Hyp-NH2 |
ADAMTS-4-2, at 25°C |
680769 |