EC Number   |
Inhibitors |
Structure |
|---|
    4.1.1.65 | 4-Bromo-3-hydroxybenzyloxyamine |
- |
   |
| 4.1.1.65 | 7-chloro-N-(4-ethoxyphenyl)-4-quinolinamine |
inhibitor with potent activity against Plasmodium falciparum, and low toxicity toward mammalian cells |
|
| 4.1.1.65 | 7-chloro-N-(4-propylphenyl)-4-quinolinamine |
0.01 mM, 29% inhibition, 0.1 mM, 76% inhibition of catalysis. Compound inhibits PSD activity and blocks Plasmodium falciparum blood stage development in the malaria murine model |
|
| 4.1.1.65 | Bile salt detergents |
inactivation by dissociating the oligomeric enzyme |
|
| 4.1.1.65 | Cu2+ |
- |
|
| 4.1.1.65 | Cyanoborohydride |
inactivation in presence of phosphatidylserine, no inactivation in absence of phosphatidylserine |
|
| 4.1.1.65 | Cyanoborohydride |
- |
|
| 4.1.1.65 | cycloserine |
- |
|
| 4.1.1.65 | D-penicillamine |
- |
|
| 4.1.1.65 | deoxypyridoxine |
reversion by pyridoxal phosphate |
|
