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Results 1 - 10 of 14 > >>
EC Number
Inhibitors
Commentary
Structure
(Z)-3-(2,5-dimethoxyphenyl)-2-(4-methoxyphenyl) acrylonitrile
potential of this inhibitor for the treatment of Staphylococcus aureus infections
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(Z)-3-(2,5-dimethoxyphenyl)-2-(4-methoxyphenyl) acrylonitrile
50% inhibition with 0.0101 mg/ml
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berberine chloride
potential of this inhibitor for the treatment of Staphylococcus aureus infections
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beta-sitosterol-3-O-glucopyranoside
potential of this inhibitor for the treatment of Staphylococcus aureus infections
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galangin
IC50 for recombinant SrtB(DELTA30): 0.03837 mM, no antibacterial activity against Staphylococcus aureus
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galangin-3-methyl ether
IC50 for recombinant SrtB(DELTA30): 0.1136 mM, no antibacterial activity against Staphylococcus aureus
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isorhamnetin
IC50 for recombinant SrtB(DELTA30): 0.04335 mM, no antibacterial activity against Staphylococcus aureus
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kaempferol
IC50 for recombinant SrtB(DELTA30): 0.02455 mM, no antibacterial activity against Staphylococcus aureus
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more
aryl (beta-amino)ethyl ketones inhibit sortase enzymes. Inhibition of sortases occurs through an irreversible, covalent modification of their active site cysteine. Sortases specifically activate this class of molecules via beta-elimination, generating a reactive olefin intermediate that covalently modifies the cysteine thiol
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morin
IC50 for recombinant SrtB(DELTA30): 0.00854 mM, no antibacterial activity against Staphylococcus aureus
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Results 1 - 10 of 14 > >>