EC Number |
Inhibitors |
Structure |
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3.4.22.53 | more |
suppression of calpain-2 expression with adenovirus vector-mediated RNAi |
|
3.4.22.53 | more |
specific capn2 shRNA reduces expression of the targeted isoform |
|
3.4.22.53 | more |
not inhibited by benzyloxycarbonyl-VAD-fluoromethylketone |
|
3.4.22.53 | more |
not inhibited by Ac-Thr-Pro-Leu-alpha-azaglycine-Ser-Pro-NH2, Ac-Pro-Leu-alpha-azaglycine-Ser-Pro-Pro-Pro-Ser-NH2, Ac-Leu-alpha-azaglycine-Ser-Pro-Pro-Pro-Ser-NH2, Ac-alpha-azaglycine-Ser-Pro-Pro-Pro-Ser-NH2, Ac-Thr-Pro-Thr-alpha-azaglycine-Ser-Pro-Pro-Pro-Ser-NH2, Ac-Thr-Pro-Leu-alpha-azaglycine-Ser-Ser-Pro-Pro-Ser-NH2, Ac-Thr-Pro-Leu-alpha-azaglycine-Ser-Gln-Pro-Pro-Ser-NH2, Ac-Thr-Pro-Val-alpha-azaglycine-Ser-Pro-Pro-Pro-Ser-NH2, Ac-Thr-Pro-Leu-alpha-azaglycine-Thr-Pro-Pro-Pro-Ser-NH2, and Ac-Thr-Pro-Leu-alpha-azaglycine-Arg-Pro-Pro-Pro-Ser-NH2 |
|
3.4.22.53 | Mg2+ |
5 mM, inhibits in presence of 5 mM Ca2+ |
|
3.4.22.53 | Mn2+ |
2.5 mM, strong |
|
3.4.22.53 | Zn2+ |
5 mM, inhibits in presence of 5 mM Ca2+ |
|
3.4.22.53 | Zn2+ |
5 mM, completely blocks activation of the enzyme by Ca2+ |
|
3.4.22.53 | Zn2+ |
5 mM |
|
3.4.22.53 | Zn2+ |
2.5 mM, complete |
|