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<< < Results 11 - 20 of 211 > >>
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EC Number Inhibitors Commentary Structure
Display the word mapDisplay the reaction diagram Show all sequences 3.4.24.82(2R)-2-[(biphenyl-4-ylsulfonyl)amino]-3-methylbutanoic acid - Go to the Ligand Summary Page
Display the word mapDisplay the reaction diagram Show all sequences 3.4.24.82(2R)-2-[[(3'-carbamoylbiphenyl-4-yl)sulfonyl]amino]-3-methylbutanoic acid - Go to the Ligand Summary Page
Display the word mapDisplay the reaction diagram Show all sequences 3.4.24.82(2R)-2-[[(3'-cyanobiphenyl-4-yl)sulfonyl]amino]-3-methylbutanoic acid - Go to the Ligand Summary Page
Display the word mapDisplay the reaction diagram Show all sequences 3.4.24.82(2R)-2-[[(3'-hydroxybiphenyl-4-yl)sulfonyl]amino]-3-methylbutanoic acid - Go to the Ligand Summary Page
Display the word mapDisplay the reaction diagram Show all sequences 3.4.24.82(2R)-2-[[(4'-hydroxybiphenyl-4-yl)sulfonyl]amino]-3-methylbutanoic acid - Go to the Ligand Summary Page
Display the word mapDisplay the reaction diagram Show all sequences 3.4.24.82(2R)-3-methyl-2-[([4'-[(methylcarbamoyl)oxy]biphenyl-4-yl]sulfonyl)amino]butanoic acid - Go to the Ligand Summary Page
Display the word mapDisplay the reaction diagram Show all sequences 3.4.24.82(2R)-N4-hydroxy-2-(3-hydroxybenzyl)-N1-[(1S,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]butanediamide - Go to the Ligand Summary Page
Display the word mapDisplay the reaction diagram Show all sequences 3.4.24.82(2R)-N4-hydroxy-2-(3-hydroxybenzyl)-N1-[(1S,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]butanediamide the reduced pattern of H-bond interactions is suitable for the flexible environment of ADAMTS4 and ADAMTS5 since it enables the inhibitor to re-optimizing its interaction pattern step-by-step, following the loop motion. The conformational flexibility observed for the S1' loop of ADAMTS4 and ADAMTS5 seems to be correlated to the motion of the TS-domain Go to the Ligand Summary Page
Display the word mapDisplay the reaction diagram Show all sequences 3.4.24.82(2R,5R)-1-([4-[(2,4-dichlorobenzyl)oxy]phenyl]sulfonyl)-N,5-dihydroxy-3,3-dimethylpiperidine-2-carboxamide - Go to the Ligand Summary Page
Display the word mapDisplay the reaction diagram Show all sequences 3.4.24.82(2R,5R)-1-([4-[(5-fluoro-2-methylbenzyl)oxy]phenyl]sulfonyl)-N,5-dihydroxypiperidine-2-carboxamide IC50: 145 nM Go to the Ligand Summary Page
<< < Results 11 - 20 of 211 > >>
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