EC Number   |
Inhibitors |
Structure |
|---|
   3.4.22.69 | N-benzyl-2-(N-(4-(tert-butyl)phenyl)-2-chloroacetamido)-2-(pyridin-3-yl)acetamide |
- |
 |
| 3.4.22.69 | N-ethyl-N-phenyldithiocarbamic acid zinc |
- |
  |
| 3.4.22.69 | N-tert-butyl-2-[2,3-dichloro-4-(2-methylidenebutanoyl)phenoxy]acetamide |
- |
|
| 3.4.22.69 | N-tert-butyl-L-seryl-L-valyl-N-[(1S,2E)-4-ethoxy-1-[[(3S)-3-methyl-2-oxopyrrolidin-3-yl]methyl]-4-oxobut-2-en-1-yl]-L-phenylalaninamide |
- |
|
| 3.4.22.69 | N-tert-butyl-L-seryl-L-valyl-N-[(1S,2E)-4-ethoxy-4-oxo-1-[2-(2-oxopyrrolidin-3-yl)ethyl]but-2-en-1-yl]-L-leucinamide |
- |
|
| 3.4.22.69 | N-[(1E)-3-[(2E)-2-(4-hydroxy-3,5-dimethoxybenzylidene)hydrazinyl]-3-oxo-1-phenylprop-1-en-2-yl]benzamide |
competitive inhibitor, 56.11% inhibition at 0.1 mM |
|
| 3.4.22.69 | N-[(1R)-2-(tert-butylamino)-2-oxo-1-(pyridin-3-yl)ethyl]-N-(4-tert-butylphenyl)furan-2-carboxamide |
- |
|
| 3.4.22.69 | N-[(1R)-2-(tert-butylamino)-2-oxo-1-(pyridin-3-yl)ethyl]-N-(4-tert-butylphenyl)furan-2-carboxamide |
noncovalent inhibitor, evaluation of unbinding pathways |
|
| 3.4.22.69 | N-[(1Z)-3-[[3-(dimethylamino)propyl]amino]-1-[5-(2-nitrophenyl)furan-2-yl]-3-oxoprop-1-en-2-yl]-4-methylbenzamide |
competitive inhibitor, 81.43% inhibition at 0.1 mM |
|
| 3.4.22.69 | N-[(1Z)-3-[[3-(dimethylamino)propyl]amino]-1-[5-(3-nitrophenyl)furan-2-yl]-3-oxoprop-1-en-2-yl]-4-methylbenzamide |
competitive inhibitor, 82.59% inhibition at 0.1 mM |
|
