3.4.23.39 0.000000001631 - N,N-dibutyl-N'-(4-pentylbenzyl)-N'-(4-pyrimidin-5-ylbenzyl)ethane-1,2-diamine IC50: 0.001631 nM 668255 3.4.23.39 0.000000003329 - N-(2-aminoethyl)-N-(biphenyl-4-ylmethyl)-4-pentylbenzamide IC50: 0.003329 nM 668255 3.4.23.39 0.0000001 - Iva-Val-Val-Sta-Ala-Sta IC50: 0.1 nM 648193 3.4.23.39 0.0000002 - pepstatin pH 5.0, temperature not specified in the publication 708121 3.4.23.39 0.0000005 - N'-(3,4-dimethylacridin-9-yl)-3-methylbenzohydrazide pH and temperature not specified in the publication 754374 3.4.23.39 0.0000006 - Ac-Val-Val-Sta-Ala-Sta IC50: 0.6 nM 648193 3.4.23.39 0.000004 - N'-(3,4-dimethylacridin-9-yl)-2-hydroxybenzohydrazide pH and temperature not specified in the publication 754374 3.4.23.39 0.0000043 - (1Z)-(3,4-dimethoxyphenyl)-N'-[[(3,4,5-trichlorophenoxy)acetyl]oxy]ethanimidamide pH and temperature not specified in the publication 754374 3.4.23.39 0.0000043 - (1Z)-N'-{[(4-chloro-3,5-dimethylphenoxy)acetyl]oxy}-2-(3,4-dimethoxyphenyl)ethanimidamide pH 4.5, 37°C 708120 3.4.23.39 0.0000043 - N-[(2S,3S)-2-hydroxy-3-[(phenoxyacetyl)amino]-4-phenylbutyl]-N-[2-(4-methoxyphenyl)ethyl]piperidine-4-carboxamide predicted inhibition constant, temperature not specified in the publication, pH not specified in the publication 717478 3.4.23.39 0.0000044 - N-(cyclopentylcarbamothioyl)-4-ethoxy-3-nitrobenzamide pH and temperature not specified in the publication 754374 3.4.23.39 0.0000045 - N-[(cyclopentylamino)carbonothioyl]-4-ethoxy-3-nitrobenzamide pH 4.5, 37°C 708120 3.4.23.39 0.0000055 - 4-amino-N'-[(2,4-dichlorobenzyl)oxy]-N-(2-methylphenyl)-1,2,5­oxadiazole-3-carboximidamide pH 4.5, 37°C 708120 3.4.23.39 0.0000055 - 4-amino-N'-[(2,4-dichlorophenyl)methoxy]-N-(2-methylphenyl)-1,2,5-oxadiazole-3-carboximidamide pH and temperature not specified in the publication 754374 3.4.23.39 0.000006 - (2R,3R,4S,6R)-6-[[(E)-2-(4-acetylphenyl)ethenyl]oxy]-2-[[(2E)-3-(4-acetylphenyl)prop-2-en-1-yl]oxy]-3,4-dihydroxy-N,N'-bis[(1S,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]heptanediamide predicted inhibition constant, temperature not specified in the publication, pH not specified in the publication 717478 3.4.23.39 0.0000064 - 4-amino-N'-(benzyloxy)-N-(2-methylphenyl)-1,2,5-oxadiazole-3-carboximidamide pH and temperature not specified in the publication 754374 3.4.23.39 0.0000064 - 4-amino-N'-(benzyloxy)-N-(2-methylphenyl)-1,2,5-oxadiazole-3­carboximidamide pH 4.5, 37°C 708120 3.4.23.39 0.0000076 - N',N'''-1,2-phenylenebis[N-(3-chlorophenyl)urea] pH 4.5, 37°C 708120 3.4.23.39 0.0000076 - N'-(4-chlorophenyl)-N'-(2-[[(3-chlorophenyl)carbamoyl]amino]phenyl)urea pH and temperature not specified in the publication 754374 3.4.23.39 0.0000088 - N-([(2,4-dimethylphenyl)amino][(4-oxo-1,4,5,6,7,8-hexahydro-2-quinazolinyl)amino]methylene)benzamide pH 4.5, 37°C 708120 3.4.23.39 0.0000088 - N-[(E)-[(2,4-dimethylphenyl)amino][(4-oxo-1,4,5,6,7,8-hexahydroquinolin-2-yl)amino]methylidene]benzamide pH and temperature not specified in the publication 754374 3.4.23.39 0.0000095 - N-(3,4-dichlorophenyl)-2-[(4,6-dimethyl-2-pyrimidinyl)amino]­3a,4,5,6,7,7a-hexahydro-1H-benzimidazole-1-carboxamide pH 4.5, 37°C 708120 3.4.23.39 0.0000095 - N-(3,4-dichlorophenyl)-2-[(4,6-dimethylpyrimidin-2-yl)amino]-3a,4,5,6,7,7a-hexahydro-1H-benzimidazole-1-carboxamide pH and temperature not specified in the publication 754374 3.4.23.39 0.00001 - N-[(2S,3S)-5-[[(2S)-1-[[(2S)-1-amino-4-methyl-1-oxopentan-2-yl]amino]-1-oxopropan-2-yl]amino]-1-[(4-bromobenzyl)oxy]-3-hydroxy-5-oxopentan-2-yl]-2,4,6-trifluorobenzamide predicted inhibition constant, temperature not specified in the publication, pH not specified in the publication 717478 3.4.23.39 0.000011 - methyl [4'-([[1-(3-methylbutyl)piperidin-4-yl][(4-pentylphenyl)carbonyl]amino]methyl)biphenyl-4-yl]acetate - 679228 3.4.23.39 0.000014 - methyl [4'-([[1-(3-methylbutyl)piperidin-4-yl][(4-pentylcyclohexyl)carbonyl]amino]methyl)biphenyl-4-yl]acetate - 679228 3.4.23.39 0.000018 - N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-N-[1-(3-methylbutyl)piperidin-4-yl]-4-pentylbenzamide pH and temperature not specified in the publication 754374 3.4.23.39 0.000018 - N-[4-(3,4-diethylisoxazol-5-yl)benzyl]-N-[1-(3-methylbutyl)piperidin-4-yl]-4-pentylbenzamide - 679228 3.4.23.39 0.000019 - N-([5-[3,5-bis(trifluoromethyl)phenyl]furan-2-yl]methyl)-N-[1-(3-methylbutyl)piperidin-4-yl]-4-pentylbenzamide pH and temperature not specified in the publication 754374 3.4.23.39 0.000019 - N-([5-[3,5-bis(trifluoromethyl)phenyl]furan-2-yl]methyl)-N-[1-(3-methylbutyl)piperidin-4-yl]-5-pentylpyridine-2-carboxamide - 679228 3.4.23.39 0.000022 - N-((S)-1-(((2S,3S)-3-hydroxy-5-oxo-5-(((S)-1-oxo-3-phenyl-1-(prop-2-yn-1-ylamino)propan-2-yl)amino)-1-phenylpentan-2-yl)-amino)-3-methyl-1-oxobutan-2-yl)picolinamide pH 5.0, 37°C 709477 3.4.23.39 0.000028 - N-((S)-1-(((2S,3S)-5-(((R)-1-(((S)-1-amino-4-methyl-1-oxopentan-2-yl)amino)-3-chloro-1-oxopropan-2-yl)amino)-3-hydroxy-5-oxo-1-phenylpentan-2-yl)amino)-3-methyl-1-oxobutan-2-yl)-picolinamide pH 5.0, 37°C 709477 3.4.23.39 0.00003 - (1R,2R,3R,4S)-3-[[4-(2-cyclopentylethyl)phenyl]sulfonyl]-N-(naphthalen-2-ylmethyl)-7-azabicyclo[2.2.1]heptan-2-amine pH and temperature not specified in the publication 754374 3.4.23.39 0.00003 - N-benzyl-2-([3-(3-nitrophenyl)acryloyl]amino)benzamide pH 4.5, 37°C 708120 3.4.23.39 0.000031 - N-([[1-(3-methylbutyl)piperidin-4-yl](4-pentylbenzoyl)amino]methyl)-1-benzothiophene-2-carboxamide pH and temperature not specified in the publication 754374 3.4.23.39 0.000031 - N-[4-([[1-(3-methylbutyl)piperidin-4-yl][(4-pentylphenyl)carbonyl]amino]methyl)phenyl]-1-benzothiophene-2-carboxamide - 679228 3.4.23.39 0.000032 - N-[4-[5-(3,4-dimethoxybenzyl)-1,2,4-oxadiazol-3-yl]benzyl]-N-[1-(3-methylbutyl)piperidin-4-yl]-4-pentylbenzamide - 679228 3.4.23.39 0.000032 - N-[[5-(3,4-dimethoxybenzyl)-1,2,4-oxadiazol-3-yl]methyl]-N-[1-(3-methylbutyl)piperidin-4-yl]-4-pentylbenzamide pH and temperature not specified in the publication 754374 3.4.23.39 0.000034 - methyl [4'-([[1-(1H-imidazol-2-ylmethyl)piperidin-4-yl](4-pentylbenzoyl)amino]methyl)biphenyl-4-yl]acetate pH and temperature not specified in the publication 754374 3.4.23.39 0.000034 - methyl [4'-([[1-(1H-imidazol-2-ylmethyl)piperidin-4-yl][(4-pentylphenyl)carbonyl]amino]methyl)biphenyl-4-yl]acetate - 679228 3.4.23.39 0.0000389 - N-(2-([3-(1,3-benzodioxol-5-yl)-3-oxo-1-propen-1-yl]amino)phenyl)-4-nitrobenzenesulfonamide pH 4.5, 37°C 708120 3.4.23.39 0.000039 - 2,3,4-trifluoro-N-([[1-(3-methylbutyl)piperidin-4-yl](4-pentylbenzoyl)amino]methyl)benzamide pH and temperature not specified in the publication 754374 3.4.23.39 0.000039 - 2,3-difluoro-4-methyl-N-[4-([[1-(3-methylbutyl)piperidin-4-yl][(4-pentylphenyl)carbonyl]amino]methyl)phenyl]benzamide - 679228 3.4.23.39 0.0000426 - 4-amino-N'-[(2-methyl-1-naphthyl)methoxy]-1,2,5-oxadiazole-3­carboximidamide pH 4.5, 37°C 708120 3.4.23.39 0.000046 - N-((4'-[2-(benzylamino)-2-oxoethyl]biphenyl-4-yl)methyl)-N-[2-(dibutylamino)ethyl]-4-pentylbenzamide IC50: 46 nM 667988 3.4.23.39 0.000047 - N-[[5-(3,4-dichlorophenyl)furan-2-yl]methyl]-N-[1-(3-methylbutyl)piperidin-4-yl]-4-pentylbenzamide - 679228 3.4.23.39 0.000047 - N-[[5-(3,4-dichlorophenyl)furan-2-yl]methyl]-N-[1-(3-methylbutyl)piperidin-4-yl]-4-pentylbenzamide pH and temperature not specified in the publication 754374 3.4.23.39 0.00005 - (1R,2R,3R,4S)-3-[(4-heptylphenyl)sulfonyl]-N-(naphthalen-2-ylmethyl)-7-azabicyclo[2.2.1]heptan-2-amine pH and temperature not specified in the publication 754374 3.4.23.39 0.00005 - (1R,2R,3R,4S)-3-[[4-(4,4-dimethylpentyl)phenyl]sulfonyl]-N-(naphthalen-2-ylmethyl)-7-azabicyclo[2.2.1]heptan-2-amine pH and temperature not specified in the publication 754374 3.4.23.39 0.000054 - N-[1-(3-methylbutyl)piperidin-4-yl]-5-pentyl-N-[[4'-(piperidin-1-ylcarbonyl)biphenyl-4-yl]methyl]pyridine-2-carboxamide - 679228 3.4.23.39 0.000054 - N-[1-(3-methylbutyl)piperidin-4-yl]-5-pentyl-N-[[4'-(piperidin-1-ylcarbonyl)biphenyl-4-yl]methyl]pyridine-2-carboxamide pH and temperature not specified in the publication 754374 3.4.23.39 0.000056 - N-[2-(dibutylamino)ethyl]-4-pentyl-N-([4'-(thiomorpholin-4-ylcarbonyl)biphenyl-4-yl]methyl)benzamide IC50: 56 nM 667988 3.4.23.39 0.000056 - N-[4-(1,3-benzodioxol-5-yl)benzyl]-N-[2-(dibutylamino)ethyl]benzamide IC50: 56 nM 668255 3.4.23.39 0.0000573 - 6-((2-[(5-chloro-2-methoxyphenyl)amino]-2-oxoethyl)thio)-5-cyano-N-(2-methoxyphenyl)-2-methyl-4-phenyl-1,4-dihydro-3-pyridinecarboxamide pH 4.5, 37°C 708120 3.4.23.39 0.0000621 - N-((2,3-dihydro-1,4-benzodioxin-6-ylamino)[(6-methyl-4-oxo-1,4-dihydro-2-pyrimidinyl)amino]methylene)benzamide pH 4.5, 37°C 708120 3.4.23.39 0.000067 - N-[[5-(2,5-dichlorophenyl)furan-2-yl]methyl]-N-[1-(3-methylbutyl)piperidin-4-yl]-4-pentylbenzamide - 679228 3.4.23.39 0.000067 - N-[[5-(2,5-dichlorophenyl)furan-2-yl]methyl]-N-[1-(3-methylbutyl)piperidin-4-yl]-4-pentylbenzamide pH and temperature not specified in the publication 754374 3.4.23.39 0.000072 - N-benzyl-4'-(([2-(dibutylamino)ethyl][(4-pentylphenyl)carbonyl]amino)methyl)biphenyl-4-carboxamide IC50: 72 nM 667988 3.4.23.39 0.000074 - N-[2-(dibutylamino)ethyl]-N-([4'-(2-morpholin-4-yl-2-oxoethyl)biphenyl-4-yl]methyl)-4-pentylbenzamide IC50: 74 nM 667988 3.4.23.39 0.000077 - 4'-(([2-(dibutylamino)ethyl][(4-pentylphenyl)carbonyl]amino)methyl)-N,N-dimethylbiphenyl-4-carboxamide IC50: 77 nM 667988 3.4.23.39 0.0000875 - N-(2-methoxyphenyl)-2-(5H-[1,2,4]triazino[5,6-b]indol-3­ylthio)butanamide pH 4.5, 37°C 708120 3.4.23.39 0.0000875 - pepstatin A pH 4.5, 37°C 708120 3.4.23.39 0.000089 - (1R,2R,3R,4S,5R)-5-[(cyclobutylamino)methyl]-N-(naphthalen-2-ylmethyl)-3-[(4-pentylphenyl)sulfonyl]-7-azabicyclo[2.2.1]heptan-2-amine pH and temperature not specified in the publication 754374 3.4.23.39 0.000091 - N-[2-(dibutylamino)ethyl]-N-([4'-(2-morpholin-4-yl-2-oxoethyl)biphenyl-4-yl]methyl)-4-pentylbenzamide IC50: 91 nM 667988 3.4.23.39 0.0000961 - 2-(1,3-benzothiazol-2-ylamino)-N-(2-chlorophenyl)-6-oxo-1,4,5,6­tetrahydro-4-pyrimidinecarboxamide pH 4.5, 37°C 708120 3.4.23.39 0.0001 - (1R,2R,3R,4S,5R)-5-[(cyclopentylamino)methyl]-N-(naphthalen-2-ylmethyl)-3-[(4-pentylphenyl)sulfonyl]-7-azabicyclo[2.2.1]heptan-2-amine pH and temperature not specified in the publication 754374 3.4.23.39 0.000101 - N-[4-(1,3-benzodioxol-5-yl)benzyl]-N-[2-(dibutylamino)ethyl]-4-pentylbenzamide IC50: 101 nM 667988 3.4.23.39 0.000104 - N-[2-(dibutylamino)ethyl]-N-([4'-(2-hydroxyethoxy)biphenyl-4-yl]methyl)benzamide IC50: 104 nM 668255 3.4.23.39 0.000112 - N-[4-(benzyloxy)benzyl]-N-[2-(dibutylamino)ethyl]-4-pentylbenzamide IC50: 112 nM 668255 3.4.23.39 0.000113 - N-[1-(3-methylbutyl)piperidin-4-yl]-N-[4-[methyl(pyridin-4-yl)amino]benzyl]-4-pentylbenzamide - 679228 3.4.23.39 0.000113 - N-[1-(3-methylbutyl)piperidin-4-yl]-N-[[methyl(pyridin-3-yl)amino]methyl]-4-pentylbenzamide pH and temperature not specified in the publication 754374 3.4.23.39 0.0001181 - N-((2,3-dihydro-1,4-benzodioxin-6-ylamino)[(6-oxo-4-propyl-1,6-dihydro-2-pyrimidinyl)amino]methylene)-4-methoxybenzamide pH 4.5, 37°C 708120 3.4.23.39 0.0001229 - N-(([6-methyl-2-(4-methylphenyl)-2H-1,2,3-benzotriazol-5-yl]amino)carbonothioyl)-2-nitrobenzamide pH 4.5, 37°C 708120 3.4.23.39 0.000124 - methyl [4'-(([2-(dibutylamino)ethyl](phenylcarbonyl)amino)methyl)biphenyl-4-yl]acetate IC50: 124 nM 668255 3.4.23.39 0.00013 - (1R,2R,3R,4S)-3-[(4-hexylphenyl)sulfonyl]-N-(naphthalen-2-ylmethyl)-7-azabicyclo[2.2.1]heptan-2-amine pH and temperature not specified in the publication 754374 3.4.23.39 0.00013 - (1S,2S,3S,4R)-3-(4-hexylphenylsulfonyl)-N-(naphthalen-2-ylmethyl)-7-azabicyclo[2.2.1]heptan-2-amine - 677552 3.4.23.39 0.000141 - N-((S)-1-(((2S,3S)-5-(((S)-1-(((S)-1-amino-4-methyl-1-oxopentan-2-yl)amino)-1-oxopent-4-yn-2-yl)amino)-3-hydroxy-5-oxo-1-phenylpentan-2-yl)amino)-3-methyl-1-oxobutan-2-yl)-picolinamide pH 5.0, 37°C 709477 3.4.23.39 0.000143 - N-(biphenyl-4-ylmethyl)-N-[2-(dibutylamino)ethyl]-4-pentylbenzamide IC50: 143 nM 667988 3.4.23.39 0.000145 - N-[1-(3-methylbutyl)piperidin-4-yl]-N-(2-[4-[methyl(2-methylquinolin-4-yl)amino]phenyl]ethyl)-4-pentylbenzamide pH and temperature not specified in the publication 754374 3.4.23.39 0.000145 - N-[1-(3-methylbutyl)piperidin-4-yl]-N-[4-[(2-methylquinolin-4-yl)amino]benzyl]-4-pentylbenzamide - 679228 3.4.23.39 0.0001452 - 2-(1-naphthyl)-N'-[(4-nitrobenzoyl)oxy]ethanimidamide pH 4.5, 37°C 708120 3.4.23.39 0.000146 - N-([[1-(3-methylbutyl)piperidin-4-yl](4-pentylbenzoyl)amino]methyl)pyridine-3-carboxamide pH and temperature not specified in the publication 754374 3.4.23.39 0.000146 - N-[1-(3-methylbutyl)piperidin-4-yl]-4-pentyl-N-[4-[(pyridin-3-ylmethyl)carbamoyl]benzyl]benzamide - 679228 3.4.23.39 0.0001464 - N-(([2-(4-ethylphenyl)-6-methyl-2H-1,2,3-benzotriazol-5-yl]amino)carbonothioyl)-2-nitrobenzamide pH 4.5, 37°C 708120 3.4.23.39 0.00015 - (1R,2R,3R,4S)-N-(naphthalen-2-ylmethyl)-3-[[4-(pentyloxy)phenyl]sulfonyl]-7-azabicyclo[2.2.1]heptan-2-amine pH and temperature not specified in the publication 754374 3.4.23.39 0.00015 - butyloxycarbonyl-His-Pro-Phe-His-Leu-PSI[CH(OH)-CH2]-Val-Ile-His IC50: 150 nM 648193 3.4.23.39 0.000151 - N-[2-(dibutylamino)ethyl]-N-([4'-(2-hydroxyethyl)biphenyl-4-yl]methyl)benzamide IC50: 151 nM 668255 3.4.23.39 0.000154 - N-[4-(([2-(dibutylamino)ethyl][(4-pentylphenyl)carbonyl]amino)methyl)phenyl]-2-methoxypyridine-4-carboxamide IC50: 154 nM 667988 3.4.23.39 0.00016 - N-[(4'-cyanobiphenyl-4-yl)methyl]-N-[2-(dibutylamino)ethyl]benzamide IC50: 160 nM 668255 3.4.23.39 0.000165 - N-[4-(1,3-benzodioxol-5-yl)benzyl]-4-pentyl-N-(2-[4-(3-phenylpropyl)piperidin-1-yl]ethyl)benzamide IC50: 165 nM 667988 3.4.23.39 0.00017 - (1R,2R,3R,4S)-3-[[4-(2-cyclobutylethyl)phenyl]sulfonyl]-N-(naphthalen-2-ylmethyl)-7-azabicyclo[2.2.1]heptan-2-amine pH and temperature not specified in the publication 754374 3.4.23.39 0.000183 - methyl [4'-(([2-(dibutylamino)ethyl][(4-pentylphenyl)carbonyl]amino)methyl)biphenyl-4-yl]acetate IC50: 183 nM 667988 3.4.23.39 0.0001871 - 2-anilino-4-(3-furyl)-6-oxo-N-phenyl-1-cyclohexene-1-carboxamide pH 4.5, 37°C 708120 3.4.23.39 0.000188 - N-[2-(dibutylamino)ethyl]-4-pentyl-N-(4-thiomorpholin-4-ylbenzyl)benzamide IC50: 188 nM 667988 3.4.23.39 0.000189 - 2-anilino-3-chloro-N-phenyl-4-(phenylimino)-2-butenamide pH 4.5, 37°C 708120 3.4.23.39 0.00019 - (1R,2R,3R,4S)-3-[[4-(3-cyclopentylpropyl)phenyl]sulfonyl]-N-(naphthalen-2-ylmethyl)-7-azabicyclo[2.2.1]heptan-2-amine pH and temperature not specified in the publication 754374 3.4.23.39 0.00019 - N-[4-(1,3-benzodioxol-5-yl)benzyl]-N-[2-(4-benzylpiperidin-1-yl)ethyl]-4-pentylbenzamide IC50: 190 nM 667988 3.4.23.39 0.000191 - N-[(2'-chlorobiphenyl-4-yl)methyl]-N-[2-(dibutylamino)ethyl]benzamide IC50: 191 nM 668255 3.4.23.39 0.000195 - N-[4-(1,3-benzodioxol-5-yl)benzyl]-N-[3-(dibutylamino)propyl]-4-pentylbenzamide IC50:195 nM 668255 3.4.23.39 0.000197 - [4'-(([2-(dibutylamino)ethyl](phenylcarbonyl)amino)methyl)biphenyl-4-yl]acetic acid IC50: 197 nM 668255 3.4.23.39 0.0002 - N-[2-(dibutylamino)ethyl]-4-pentyl-N-[4-(4-phenylpiperazin-1-yl)benzyl]benzamide IC50: 200 nM 667988 3.4.23.39 0.0002011 - 3-chloro-N-([2-(2-methoxybenzoyl)hydrazino]carbonothioyl)-1-benzothiophene-2-carboxamide pH 4.5, 37°C 708120 3.4.23.39 0.000202 - N-[4-(([2-(dibutylamino)ethyl][(4-pentylphenyl)carbonyl]amino)methyl)phenyl]piperidine-3-carboxamide IC50: 202 nM 667988 3.4.23.39 0.000204 - N-[2-(dibutylamino)ethyl]-N-(4-pyrimidin-5-ylbenzyl)benzamide IC50: 204 nM 668255 3.4.23.39 0.000208 - 4'-(([2-(dibutylamino)ethyl](phenylcarbonyl)amino)methyl)biphenyl-3-carboxylic acid IC50: 208 nM 668255 3.4.23.39 0.00021 - (1S,2S,3S,4R)-N-(3-bromobenzyl)-3-(4-hexylphenylsulfonyl)-7-azabicyclo[2.2.1]heptan-2-amine - 677552 3.4.23.39 0.000212 - N-[2-(dibutylamino)ethyl]-4-pentyl-N-(4-pyridin-4-ylbenzyl)benzamide IC50: 212 nM 667988 3.4.23.39 0.000221 - N-[3-(dibutylamino)propyl]-4-pentyl-N-([4'-(2-pyrrolidin-1-ylethoxy)biphenyl-4-yl]methyl)benzamide IC50: 221 nM 668255 3.4.23.39 0.000224 - N-[2-(dibutylamino)ethyl]-4-pentyl-N-[4-(phenylamino)benzyl]benzamide IC50: 224 nM 667988 3.4.23.39 0.000236 - N-[[5-(4-chlorophenyl)-1,2-oxazol-3-yl]methyl]-N-[1-(3-methylbutyl)piperidin-4-yl]-4-pentylbenzamide pH and temperature not specified in the publication 754374 3.4.23.39 0.000236 - N-[[5-(4-chlorophenyl)isoxazol-3-yl]methyl]-N-[1-(3-methylbutyl)piperidin-4-yl]-4-pentylbenzamide - 679228 3.4.23.39 0.0002364 - N'-[(4-methoxy-3-nitrobenzoyl)oxy]-2-(1-naphthyl)ethanimidamide pH 4.5, 37°C 708120 3.4.23.39 0.0002374 - N,N'-([(4,6-dimethyl-2-quinazolinyl)amino]methylylidene)dipropanamide pH 4.5, 37°C 708120 3.4.23.39 0.00024 - N-[2-(dibutylamino)ethyl]-4-pentyl-N-[4-(1H-pyrrol-1-yl)benzyl]benzamide IC50: 240 nM 667988 3.4.23.39 0.000243 - N-[4-(([2-(dibutylamino)ethyl][(4-pentylphenyl)carbonyl]amino)methyl)phenyl]pyrazine-2-carboxamide IC50: 243 nM 667988 3.4.23.39 0.000246 - N-[3-(dibutylamino)propyl]-N-[(4'-methoxybiphenyl-4-yl)methyl]-4-pentylbenzamide IC50: 246 nM 668255 3.4.23.39 0.000252 - N-(biphenyl-4-ylmethyl)-N-[2-(dibutylamino)ethyl]-4-pentylbenzamide IC50: 252 nM 668255 3.4.23.39 0.000284 - (1R,2R,3R,4S,6R)-6-[(cyclobutylamino)methyl]-N-(naphthalen-2-ylmethyl)-3-[(4-pentylphenyl)sulfonyl]-7-azabicyclo[2.2.1]heptan-2-amine pH and temperature not specified in the publication 754374 3.4.23.39 0.000289 - (1R,2R,3R,4S,6R)-6-[(cyclopentylamino)methyl]-N-(naphthalen-2-ylmethyl)-3-[(4-pentylphenyl)sulfonyl]-7-azabicyclo[2.2.1]heptan-2-amine pH and temperature not specified in the publication 754374 3.4.23.39 0.000289 - N-(4-[benzyl(methyl)amino]benzyl)-N-[2-(dibutylamino)ethyl]-4-pentylbenzamide IC50: 289 nM 667988 3.4.23.39 0.000293 - N-[2-(dibutylamino)ethyl]-N-[(3'-methylbiphenyl-4-yl)methyl]benzamide IC50: 293 nM 668255 3.4.23.39 0.000295 - N-[2-(dibutylamino)ethyl]-N-(4-pyridin-4-ylbenzyl)benzamide IC50: 295 nM 668255 3.4.23.39 0.000305 - 4-amino-N'-(benzyloxy)-N-(4-methylphenyl)-1,2,5-oxadiazole-3­carboximidamide pH 4.5, 37°C 708120 3.4.23.39 0.000322 - N-[3-(dibutylamino)propyl]-N-[(2'-methoxybiphenyl-4-yl)methyl]-4-pentylbenzamide IC50: 322 nM 668255 3.4.23.39 0.000333 - N-((S)-1-(((2S,3S)-5-(((S)-1-(((S)-1-amino-4-methyl-1-oxopentan-2-yl)amino)-3-cyano-1-oxopropan-2-yl)amino)-3-hydroxy-5-oxo-1-phenylpentan-2-yl)amino)-3-methyl-1-oxobutan-2-yl)picolinamide pH 5.0, 37°C 709477 3.4.23.39 0.000334 - N-[4-(1,3-benzodioxol-5-yl)benzyl]-4-pentyl-N-(2-piperidin-1-ylethyl)benzamide IC50: 334 nM 667988 3.4.23.39 0.000334 - N-[4-(1,3-benzodioxol-5-yl)benzyl]-N-(2-[benzyl(2-hydroxyethyl)amino]ethyl)-4-pentylbenzamide IC50: 334 nM 667988 3.4.23.39 0.0003467 - SC-50083 IC50: 0.0003467 mM 648187 3.4.23.39 0.00035 - (1R,2R,3R,4S)-3-[[4-(6-fluorohexyl)phenyl]sulfonyl]-N-(naphthalen-2-ylmethyl)-7-azabicyclo[2.2.1]heptan-2-amine pH and temperature not specified in the publication 754374 3.4.23.39 0.000351 - N-[2-(dibutylamino)ethyl]-N-(4-pyrimidin-5-ylbenzyl)benzamide IC50: 351 nM 668255 3.4.23.39 0.000369 - N-[2-(dibutylamino)ethyl]-4-pentyl-N-(4-piperidin-1-ylbenzyl)benzamide IC50: 369 nM 667988 3.4.23.39 0.000374 - N-[2-(dibutylamino)ethyl]-4-pentyl-N-(4-pyridin-3-ylbenzyl)benzamide IC50: 374 nM 667988 3.4.23.39 0.00038 - (1R,2R,3R,4S)-3-[[4-(3-cyclohexylpropyl)phenyl]sulfonyl]-N-(naphthalen-2-ylmethyl)-7-azabicyclo[2.2.1]heptan-2-amine pH and temperature not specified in the publication 754374 3.4.23.39 0.00038 - N-[2-(dibutylamino)ethyl]-4-pentyl-N-(4-pyridin-2-ylbenzyl)benzamide IC50: 380 nM 667988 3.4.23.39 0.00039 - (1S,2S,3S,4R)-3-(4-hexylphenylsulfonyl)-N-((2'-methoxybiphenyl-3-yl)methyl)-7-azabicyclo[2.2.1]heptan-2-amine - 677552 3.4.23.39 0.00039 - N-[2-(dibutylamino)ethyl]-N-([3'-(trifluoromethyl)biphenyl-4-yl]methyl)benzamide IC50: 390 nM 668255 3.4.23.39 0.0004 - 3'-(((1S,2S,3S,4R)-3-(4-hexylphenylsulfonyl)-7-azabicyclo[2.2.1]heptan-2-ylamino)methyl)biphenyl-2-ol - 677552 3.4.23.39 0.000407 - N-[(4'-chlorobiphenyl-4-yl)methyl]-N-[3-(dibutylamino)propyl]-4-pentylbenzamide IC50: 407 nM 668255 3.4.23.39 0.000428 - N-[2-(dibutylamino)ethyl]-N-[(3',4'-dimethoxybiphenyl-4-yl)methyl]benzamide IC50: 428 nM 668255 3.4.23.39 0.000429 - N-[4-(benzylamino)benzyl]-N-[2-(dibutylamino)ethyl]-4-pentylbenzamide IC50: 429 nM 667988 3.4.23.39 0.000437 - N-(4-[6-(1,3-benzodioxol-5-yl)pyridin-3-yl]benzyl)-N-[2-(dibutylamino)ethyl]-4-pentylbenzamide IC50: 437 nM 667988 3.4.23.39 0.000439 - N-[4-(1,3-benzodioxol-5-yl)benzyl]-N-(2-([2-(diethylamino)ethyl](ethyl)amino)ethyl)-4-pentylbenzamide IC50: 439 nM 667988 3.4.23.39 0.000441 - 2-([4'-(([2-(dibutylamino)ethyl](4-pentylbenzyl)amino)methyl)biphenyl-4-yl]oxy)ethanol IC50: 441 nM 668255 3.4.23.39 0.000446 - N-[(4'-chlorobiphenyl-4-yl)methyl]-N-[2-(dibutylamino)ethyl]benzamide IC50: 446 nM 668255 3.4.23.39 0.000463 - [4'-(([2-(dibutylamino)ethyl][(4-pentylphenyl)carbonyl]amino)methyl)biphenyl-4-yl]acetic acid IC50: 463 nM 667988 3.4.23.39 0.000464 - N-[4-(([2-(dibutylamino)ethyl][(4-pentylphenyl)carbonyl]amino)methyl)phenyl]piperidine-4-carboxamide IC50: 464 nM 667988 3.4.23.39 0.000468 - N-[3-(dibutylamino)propyl]-N-[(3',4'-dimethoxybiphenyl-4-yl)methyl]-4-pentylbenzamide IC50: 468 nM 668255 3.4.23.39 0.000469 - N-[2-(dibutylamino)ethyl]-4-pentyl-N-(3-phenoxybenzyl)benzamide IC50: 469 nM 668255 3.4.23.39 0.000495 - 4'-(([2-(dibutylamino)ethyl](phenylcarbonyl)amino)methyl)biphenyl-4-carboxylic acid IC50: 495 nM 668255 3.4.23.39 0.0005 - (5-[[(4-bromobenzoyl)oxy]methyl]-2,3,4,7-tetrahydro-1H-azepin-3-yl)methyl 4-aminobenzoate pH and temperature not specified in the publication 754374 3.4.23.39 0.000511 - N-[2-(dibutylamino)ethyl]-N-([4'-(2-hydroxyethoxy)biphenyl-4-yl]methyl)-4-pentylbenzamide IC50: 511 nM 667988 3.4.23.39 0.000531 - N-[2-(dibutylamino)ethyl]-4-pentyl-N-(4-pyrimidin-5-ylbenzyl)benzamide IC50: 531 nM 667988 3.4.23.39 0.000531 - N-[4-(1,3-benzodioxol-5-yl)benzyl]-N-[2-(dipropylamino)ethyl]-4-pentylbenzamide IC50: 531 nM 667988 3.4.23.39 0.00055 - N,N'-(3S,4S)-pyrrolidine-3,4-diylbis(N-benzyl-2-phenylacetamide) pH and temperature not specified in the publication 754374 3.4.23.39 0.000574 - N-[2-(dibutylamino)ethyl]-N-(4-[methyl(phenyl)amino]benzyl)-4-pentylbenzamide IC50: 574 nM 667988 3.4.23.39 0.00058 - N-[3-(dibutylamino)propyl]-N-[(3'-methoxybiphenyl-4-yl)methyl]-4-pentylbenzamide IC50: 580 nM 668255 3.4.23.39 0.000587 - N-[4-(2,2'-bipyridin-5-yl)benzyl]-N-[2-(dibutylamino)ethyl]-4-pentylbenzamide IC50: 587 nM 667988 3.4.23.39 0.000589 - N-[2-(dibutylamino)ethyl]-4-pentyl-N-[4-(6-phenylpyridin-3-yl)benzyl]benzamide IC50: 589 nM 667988 3.4.23.39 0.000591 - N-[(4'-butylbiphenyl-4-yl)methyl]-N-[2-(dibutylamino)ethyl]benzamide IC50: 591 nM 668255 3.4.23.39 0.000596 - N-[2-(dibutylamino)ethyl]-4-pentyl-N-[4-(trifluoromethyl)benzyl]benzamide IC50: 596 nM 668255 3.4.23.39 0.000597 - N-[3-(dibutylamino)propyl]-N-[(2'-methylbiphenyl-4-yl)methyl]-4-pentylbenzamide IC50: 597 nM 668255 3.4.23.39 0.00064 - N-benzyl-2-bromo-N-[[4-([[3-(2,4-dichlorophenyl)propyl][2-(1,3-dioxo-1,3-dihydro-2H-isoindol-2-yl)ethyl]amino]methyl)pyrrolidin-3-yl]methyl]-4,5-dimethoxybenzamide pH and temperature not specified in the publication 754374 3.4.23.39 0.000642 - N-[4-(2,4'-bipyridin-5-yl)benzyl]-N-[2-(dibutylamino)ethyl]-4-pentylbenzamide IC50: 642 nM 667988 3.4.23.39 0.000646 - N-[4-(4-benzylpiperazin-1-yl)benzyl]-N-[2-(dibutylamino)ethyl]-4-pentylbenzamide IC50: 646 nM 667988 3.4.23.39 0.00067 - N-[2-(dibutylamino)ethyl]-N-[4-(1H-indol-1-yl)benzyl]-4-pentylbenzamide IC50: 670 nM 667988 3.4.23.39 0.00068 - (1R,2R,3R,4S)-N-(naphthalen-2-ylmethyl)-3-[(4-pentylphenyl)sulfonyl]-7-azabicyclo[2.2.1]heptan-2-amine pH and temperature not specified in the publication 754374 3.4.23.39 0.000713 - 4'-(([2-(dibutylamino)ethyl](4-pentylbenzyl)amino)methyl)biphenyl-4-carbonitrile IC50: 713 nM 668255 3.4.23.39 0.000736 - N-[4-(2,2'-bipyridin-5-yl)benzyl]-N-[2-(dibutylamino)ethyl]-4-pentylbenzamide IC50: 736 nM 667988 3.4.23.39 0.00079 - 6-[4-([(1S,2R,3R,4R)-3-[(naphthalen-2-ylmethyl)amino]-7-azabicyclo[2.2.1]hept-2-yl]sulfonyl)phenyl]hexan-1-ol pH and temperature not specified in the publication 754374 3.4.23.39 0.00081 - N-benzyl-2-bromo-N-[[4-([[3-(2,4-dichlorophenyl)propyl](3-phenylpropyl)amino]methyl)pyrrolidin-3-yl]methyl]-4,5-dimethoxybenzamide pH and temperature not specified in the publication 754374 3.4.23.39 0.000831 - N-[4-(1,3-benzodioxol-5-yl)benzyl]-N',N'-dibutyl-N-(4-pentylbenzyl)ethane-1,2-diamine IC50: 831 nM 668255 3.4.23.39 0.000845 - N-[4-(benzyloxy)benzyl]-N',N'-dibutyl-N-(4-pentylbenzyl)ethane-1,2-diamine IC50: 845 nM 668255 3.4.23.39 0.0009 - (1R,2R,3R,4S)-N-(naphthalen-2-ylmethyl)-3-[[4-(2-propoxyethyl)phenyl]sulfonyl]-7-azabicyclo[2.2.1]heptan-2-amine pH and temperature not specified in the publication 754374 3.4.23.39 0.000918 - 4'-(([2-(dibutylamino)ethyl](4-pentylbenzyl)amino)methyl)biphenyl-4-carbonitrile IC50: 918 nM 668255 3.4.23.39 0.001 - 2-nitrobenzohydrazide pH and temperature not specified in the publication 754374 3.4.23.39 0.001 - butyloxycarbonyl-His-Pro-Phe-His-Sta-Leu-Phe-NH2 IC50: 1000 nM 648193 3.4.23.39 0.001022 - N,N-dibutyl-N'-[(2'-fluorobiphenyl-4-yl)methyl]-N'-(4-pentylbenzyl)ethane-1,2-diamine IC50: 0.001022 mM 668255 3.4.23.39 0.00105 - 1,2-diphenylhydrazine pH and temperature not specified in the publication 754374 3.4.23.39 0.001088 - N-(3,4-dimethylphenyl)-N'-(imino[(4,6,7-trimethyl-2-quinazolinyl)amino]methyl)thiourea pH 4.5, 37°C 708120 3.4.23.39 0.0011 - N-[3-(dibutylamino)propyl]-N-[(2'-methoxybiphenyl-4-yl)methyl]-4-pentylbenzamide IC50: 0.0011 mM 668255 3.4.23.39 0.001161 - N-(biphenyl-4-ylmethyl)-N-[2-(butylamino)ethyl]-4-pentylbenzamide IC50: 0.001161 mM 668255 3.4.23.39 0.00119 - N-([3',5'-bis(trifluoromethyl)biphenyl-4-yl]methyl)-N-[3-(dibutylamino)propyl]-4-pentylbenzamide IC50: 0.00119 mM 668255 3.4.23.39 0.00125 - butanehydrazide pH and temperature not specified in the publication 754374 3.4.23.39 0.0013 - (3S,4S)-pyrrolidine-3,4-diyl bis(naphthalen-1-ylacetate) pH and temperature not specified in the publication 754374 3.4.23.39 0.0013 - N,N-dibutyl-N'-(4-pentylbenzyl)-N'-(4-pyridin-2-ylbenzyl)ethane-1,2-diamine IC50: 0.0013 mM 668255 3.4.23.39 0.0013 - N-[4-(benzyloxy)benzyl]-4-butyl-N-[2-(dibutylamino)ethyl]benzamide IC50: 0.0013 mM 668255 3.4.23.39 0.00145 - 4,4'-(hydrazine-1,2-diyl)dipyridine pH and temperature not specified in the publication 754374 3.4.23.39 0.00147 - 2-[4'-(([2-(dibutylamino)ethyl](4-pentylbenzyl)amino)methyl)biphenyl-4-yl]ethanol IC50: 0.00147 mM 668255 3.4.23.39 0.001491 - N-[2-(dibutylamino)ethyl]-N-[4-(diethylamino)benzyl]-4-pentylbenzamide IC50: 1491 nM 667988 3.4.23.39 0.0015 - N-(biphenyl-4-ylmethyl)-4-butyl-N-[2-(dibutylamino)ethyl]benzamide IC50: 0.0015 mM 668255 3.4.23.39 0.001501 - N-[4-(1,3-benzodioxol-5-yl)benzyl]-N-(2-[bis(1-methylethyl)amino]ethyl)-4-pentylbenzamide IC50: 1501 nM 667988 3.4.23.39 0.001519 - N-[4-(1,3-benzodioxol-5-yl)benzyl]-N-[2-(diethylamino)ethyl]-4-pentylbenzamide IC50: 1519 nM 667988 3.4.23.39 0.0016 - 2,2-diphenylacetohydrazide pH and temperature not specified in the publication 754374 3.4.23.39 0.001603 - N,N-dibutyl-N'-(4-pentylbenzyl)-N'-(4-pyridin-4-ylbenzyl)ethane-1,2-diamine IC50: 0.001603 mM 668255 3.4.23.39 0.00165 - 2-methoxybenzohydrazide pH and temperature not specified in the publication 754374 3.4.23.39 0.0017 - N-([3',5'-bis(trifluoromethyl)biphenyl-4-yl]methyl)-N-[2-(dibutylamino)ethyl]benzamide IC50: 0.0017 mM 668255 3.4.23.39 0.001816 - N-[2-(dibutylamino)ethyl]-4-pentyl-N-[4-(pyridin-4-ylamino)benzyl]benzamide IC50: 1816 nM 667988 3.4.23.39 0.001831 - 6-bromo-2,3,4,9-tetrahydro-1H-carbazol-1-one N­phenylthiosemicarbazone pH 4.5, 37°C 708120 3.4.23.39 0.001912 - N-(4-[5-(1,3-benzodioxol-5-yl)pyridin-2-yl]benzyl)-N-[2-(dibutylamino)ethyl]-4-pentylbenzamide IC50: 1912 nM 667988 3.4.23.39 0.002 - (1R,4S)-6-[3-[(6-chloro-1,3-benzothiazol-2-yl)sulfanyl]propyl]-7-(naphthalen-1-ylmethoxy)-1,2,3,4-tetrahydro-1,4-epiminonaphthalene pH and temperature not specified in the publication 754374 3.4.23.39 0.002 - 1-[3-chloro-6-(trifluoromethyl)phenanthren-9-yl]-3-(dibutylamino)propan-1-ol pH and temperature not specified in the publication 754374 3.4.23.39 0.002 - N,N-dibutyl-N'-(4-pentylbenzyl)-N'-([4'-(2-pyrrolidin-1-ylethoxy)biphenyl-4-yl]methyl)ethane-1,2-diamine IC50: 0.002 mM 668255 3.4.23.39 0.002 - N-butyl-N-[2-[6-chloro-3-(3,4-dichlorophenyl)naphthalen-1-yl]-2-hydroxyethyl]butan-1-aminium pH 5.0, temperature not specified in the publication 708121 3.4.23.39 0.002 - N-[3-[1,3-dichloro-6-(trifluoromethyl)phenanthren-9-yl]-3-hydroxypropyl]-N-pentylpentan-1-aminium pH 5.0, temperature not specified in the publication 708121 3.4.23.39 0.002067 - N-(biphenyl-4-ylmethyl)-N',N'-dibutyl-N-(4-pentylbenzyl)ethane-1,2-diamine IC50: 0.002067 mM 668255 3.4.23.39 0.00221 - (1R,2R,3R,4S)-3-[[4-(4-fluorobutyl)phenyl]sulfonyl]-N-(naphthalen-2-ylmethyl)-7-azabicyclo[2.2.1]heptan-2-amine pH and temperature not specified in the publication 754374 3.4.23.39 0.002229 - N-[2-(dibutylamino)ethyl]-4-pentyl-N-[4-(6-pyrimidin-5-ylpyridin-3-yl)benzyl]benzamide IC50: 2229 nM 667988 3.4.23.39 0.0023 - 4-butyl-N-[2-(dibutylamino)ethyl]-N-(3-phenoxybenzyl)benzamide IC50: 0.0023 mM 668255 3.4.23.39 0.002317 - N-(biphenyl-4-ylmethyl)-N-[2-(diethylamino)ethyl]-4-pentylbenzamide IC50: 0.002317 mM 668255 3.4.23.39 0.002345 - N-[2-(dibutylamino)ethyl]-4-pentyl-N-[4-(5-phenylpyridin-2-yl)benzyl]benzamide IC50: 2345 nM 667988 3.4.23.39 0.002547 - N-[2-(dibutylamino)ethyl]-N-[4-(4-methylpiperazin-1-yl)benzyl]-4-pentylbenzamide IC50: 2547 nM 667988 3.4.23.39 0.002897 - N-[4-(1,3-benzodioxol-5-yl)benzyl]-N-(2-morpholin-4-ylethyl)-4-pentylbenzamide IC50: 2897 nM 667988 3.4.23.39 0.003 - (1R,4S)-6-[2-[(6-chloro-1,3-benzothiazol-2-yl)sulfanyl]ethoxy]-7-[2-(naphthalen-1-yl)ethoxy]-1,2,3,4-tetrahydro-1,4-epiminonaphthalene pH and temperature not specified in the publication 754374 3.4.23.39 0.003015 - N-[2-(dibutylamino)ethyl]-N-(4-[methyl(pyridin-4-yl)amino]benzyl)-4-pentylbenzamide IC50: 3015 nM 667988 3.4.23.39 0.0034 - N-[4-(benzyloxy)benzyl]-4-butoxy-N-[2-(dibutylamino)ethyl]benzamide IC50: 0.0034 mM 668255 3.4.23.39 0.0039 - 4-butyl-N-[2-(dibutylamino)ethyl]-N-[4-(trifluoromethyl)benzyl]benzamide IC50: 0.0039 mM 668255 3.4.23.39 0.003943 - N-(biphenyl-4-ylmethyl)-N-(2-[bis(1-methylethyl)amino]ethyl)-4-pentylbenzamide IC50: 0.003943 mM 668255 3.4.23.39 0.004 - (1R,4S)-6-[2-[(6-chloro-1,3-benzothiazol-2-yl)sulfanyl]ethoxy]-7-(naphthalen-2-ylmethoxy)-1,2,3,4-tetrahydro-1,4-epiminonaphthalene pH and temperature not specified in the publication 754374 3.4.23.39 0.004 - (1R,4S)-6-[3-(1,3-benzothiazol-2-ylsulfanyl)propyl]-7-(naphthalen-1-ylmethoxy)-1,2,3,4-tetrahydro-1,4-epiminonaphthalene pH and temperature not specified in the publication 754374 3.4.23.39 0.00419 - (1R,2R,3R,4S)-3-[(4-butylphenyl)sulfonyl]-N-(naphthalen-2-ylmethyl)-7-azabicyclo[2.2.1]heptan-2-amine pH and temperature not specified in the publication 754374 3.4.23.39 0.004553 - N-[4-(3,4'-bipyridin-6-yl)benzyl]-N-[2-(dibutylamino)ethyl]-4-pentylbenzamide IC50: 4553 nM 667988 3.4.23.39 0.00461 - 5-[4-([(1S,2R,3R,4R)-3-[(naphthalen-2-ylmethyl)amino]-7-azabicyclo[2.2.1]hept-2-yl]sulfonyl)phenyl]pentan-1-ol pH and temperature not specified in the publication 754374 3.4.23.39 0.00462 - N',N''-[1,10-phenanthroline-2,9-diyldi(E)methylylidene]bis[N-(2-methylphenyl)pyridine-2-carbohydrazonamide] pH and temperature not specified in the publication 754374 3.4.23.39 0.0047 - N-(biphenyl-4-ylmethyl)-4-butoxy-N-[2-(dibutylamino)ethyl]benzamide IC50: 0.0047 mM 668255 3.4.23.39 0.005 - (1R,4S)-6-[2-[(6-chloro-1,3-benzothiazol-2-yl)sulfanyl]ethoxy]-7-(naphthalen-1-ylmethoxy)-1,2,3,4-tetrahydro-1,4-epiminonaphthalene pH and temperature not specified in the publication 754374 3.4.23.39 0.005 - 1-[6-chloro-3-(3,4-dichlorophenyl)naphthalen-1-yl]-2-(dibutylamino)ethanol pH and temperature not specified in the publication 754374 3.4.23.39 0.005 - 2-(dihexylamino)-1-(1,2,3,4-tetrahydrophenanthren-9-yl)ethanol pH and temperature not specified in the publication 754374 3.4.23.39 0.005 - 2-[bis(4-methylpentyl)amino]-1-(1,2,3,4-tetrahydrophenanthren-9-yl)ethanol pH and temperature not specified in the publication 754374 3.4.23.39 0.005 - N-hexyl-N-[2-hydroxy-2-(1,2,3,4-tetrahydrophenanthren-9-yl)ethyl]hexan-1-aminium pH 5.0, temperature not specified in the publication 708121 3.4.23.39 0.005 - N-[2-hydroxy-2-(1,2,3,4-tetrahydrophenanthren-9-yl)ethyl]-4-methyl-N-(4-methylpentyl)pentan-1-aminium pH 5.0, temperature not specified in the publication 708121 3.4.23.39 0.005266 - N-[4-(3,3'-bipyridin-6-yl)benzyl]-N-[2-(dibutylamino)ethyl]-4-pentylbenzamide IC50: 5266 nM 667988 3.4.23.39 0.0059 - 4-butoxy-N-[2-(dibutylamino)ethyl]-N-(3-phenoxybenzyl)benzamide IC50: 0.0059 mM 668255 3.4.23.39 0.006 - [5-[(benzoyloxy)methyl]-2,3,4,7-tetrahydro-1H-azepin-3-yl]methyl 4-aminobenzoate pH and temperature not specified in the publication 754374 3.4.23.39 0.00645 - 2-[(Z)-1-(4-chlorophenyl)-2-[3-(pyridin-2-yl)isoquinolin-1-yl]ethenyl]hydrazine-1-carboximidothioic acid pH and temperature not specified in the publication 754374 3.4.23.39 0.007 - 4-methyl-N-[2-[2-(naphthalen-2-yl)hydrazinyl]phenyl]benzene-1-sulfonamide pH and temperature not specified in the publication 754374 3.4.23.39 0.007 - N-([(1RS)-3,3-difluoro-4-oxocyclohexyl]methyl)-2-(2-naphthyl)-N-(4-pentylphenyl)acetamide pH 5.0, 37°C 710185 3.4.23.39 0.007 - N-[[(1S)-3,3-difluoro-4,4-dihydroxycyclohexyl]methyl]-N-(4-pentylphenyl)naphthalene-2-carboxamide pH and temperature not specified in the publication 754374 3.4.23.39 0.00853 - N-[2-(dibutylamino)ethyl]-4-pentyl-N-[4-(5-pyrimidin-5-ylpyridin-2-yl)benzyl]benzamide IC50: 8530 nM 667988 3.4.23.39 0.0089 - N-[4-(benzyloxy)benzyl]-N-[2-(dibutylamino)ethyl]-4-propylbenzamide IC50: 0.0089 mM 668255 3.4.23.39 0.00899 - N2-(3-bromophenyl)-N-[4-[(phenylsulfanyl)methyl]phenyl]-N2-(phenylsulfonyl)glycinamide pH and temperature not specified in the publication 754374 3.4.23.39 0.009 - 2-([2-[4-([[(1S,2S,3R,4R)-3-(naphthalen-2-ylmethoxy)-7-azabicyclo[2.2.1]hept-2-yl]oxy]methyl)phenoxy]ethyl]sulfanyl)-1,3-benzothiazole pH and temperature not specified in the publication 754374 3.4.23.39 0.00947 - 1-(benzylamino)-3-(3,6-dichloro-9H-carbazol-9-yl)propan-2-ol pH and temperature not specified in the publication 754374 3.4.23.39 0.01 - (1R,4S)-6-[2-(1,3-benzothiazol-2-ylsulfanyl)ethoxy]-7-(naphthalen-2-ylmethoxy)-1,2,3,4-tetrahydro-1,4-epiminonaphthalene pH and temperature not specified in the publication 754374 3.4.23.39 0.01 - (1RS) 3,3-difluoro-N-[2-(2-naphthyl)ethyl]-4-oxo-N-(4-pentylphenyl)cyclohexanecarboxamide pH 5.0, 37°C 710185 3.4.23.39 0.01 - (1S)-3,3-difluoro-4,4-dihydroxy-N-(naphthalen-2-ylmethyl)-N-(4-pentylphenyl)cyclohexanecarboxamide pH and temperature not specified in the publication 754374 3.4.23.39 0.0103 - 4-butoxy-N-[2-(dibutylamino)ethyl]-N-[4-(trifluoromethyl)benzyl]benzamide IC50: 0.0103 mM 668255 3.4.23.39 0.0129 - N-(biphenyl-4-ylmethyl)-N-[2-(dibutylamino)ethyl]-4-propylbenzamide IC50: 0.0129 mM 668255 3.4.23.39 0.013 - (1R,4S)-6-[2-(1,3-benzothiazol-2-ylsulfanyl)ethoxy]-7-[2-(naphthalen-1-yl)ethoxy]-1,2,3,4-tetrahydro-1,4-epiminonaphthalene pH and temperature not specified in the publication 754374 3.4.23.39 0.013 - N-(4-hexylphenyl)-2-(2-naphthyl)-N-piperidin-4-ylacetamide hydrochloride pH 5.0, 37°C 710185 3.4.23.39 0.014 - (1R,4S)-6-[2-(1,3-benzothiazol-2-ylsulfanyl)ethoxy]-7-(naphthalen-1-ylmethoxy)-1,2,3,4-tetrahydro-1,4-epiminonaphthalene pH and temperature not specified in the publication 754374 3.4.23.39 0.014 - LCu(CH3COO)2 pH 4.7, 37°C 709167 3.4.23.39 0.0147 - 1-(biphenyl-4-yl)-2-[2-(pyridin-2-yl)-1H-benzimidazol-1-yl]ethanone pH 5.0, temperature not specified in the publication 717364 3.4.23.39 0.0148 - (1S,2S,3S,4R)-3-(4-bromophenylsulfonyl)-N-(naphthalen-2-ylmethyl)-7-azabicyclo[2.2.1]heptan-2-amine - 677552 3.4.23.39 0.0159 - N-[2-(dibutylamino)ethyl]-N-(3-phenoxybenzyl)-4-propylbenzamide IC50: 0.0159 mM 668255 3.4.23.39 0.016 - N-([(1RS,4SR)-3,3-difluoro-4-hydroxycyclohexyl]methyl)-2-(2-naphthyl)-N-(4-pentylphenyl)acetamide pH 5.0, 37°C 710185 3.4.23.39 0.017 - LCuCl2 pH 4.7, 37°C 709167 3.4.23.39 0.017 - N-hexyl-N-[2-hydroxy-2-(phenanthren-9-yl)ethyl]hexan-1-aminium pH 5.0, temperature not specified in the publication 708121 3.4.23.39 0.018 - 3,5,12-trihydroxy-3-(hydroxyacetyl)-10-methoxy-6,11-dioxo-1,2,3,4,5a,6,11,11a-octahydrotetracen-1-yl 3,4-di-O-acetyl-2,6-dideoxyhexopyranoside pH 5.0, temperature not specified in the publication 708121 3.4.23.39 0.019 - 2-(2-naphthyl)-N-(4-pentylphenyl)-N-piperidin-4-ylacetamide hydrochloride pH 5.0, 37°C 710185 3.4.23.39 0.019 - N-([(1RS,4RS)-3,3-difluoro-4-hydroxycyclohexyl]methyl)-2-(2-naphthyl)-N-(4-pentylphenyl)acetamide pH 5.0, 37°C 710185 3.4.23.39 0.019 - N-[2-hydroxy-2-(1,2,3,4-tetrahydrophenanthren-9-yl)ethyl]-N-pentylpentan-1-aminium pH 5.0, temperature not specified in the publication 708121 3.4.23.39 0.02 - 1-[2-hydroxy-3-(1,2,3,4,5,6,7,8-octahydrophenanthren-9-yloxy)propyl]-4-(3-methoxyphenyl)piperazin-1-ium pH 5.0, temperature not specified in the publication 708121 3.4.23.39 0.02 - N-[(1SR,3SR)-4,4-difluoro-3-hydroxycyclohexyl]-2-(2-naphthyl)-N-(4-pentylphenyl)acetamide pH 5.0, 37°C 710185 3.4.23.39 0.0212 - 1-(4-chlorophenyl)-2-[2-(pyridin-2-yl)-1H-benzimidazol-1-yl]ethanone pH 5.0, temperature not specified in the publication 717364 3.4.23.39 0.02158 - (2R,3R,4R,5R)-2,5-bis(benzyloxy)-3,4-dihydroxy-N,N'-bis[(1S,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]hexanediamide - 679228 3.4.23.39 0.024 - N-[(1SR,3RS)-4,4-difluoro-3-hydroxycyclohexyl]-2-(2-naphthyl)-N-(4-pentylphenyl)acetamide pH 5.0, 37°C 710185 3.4.23.39 0.024 - N-[3-(2,7-dichloro-9H-fluoren-4-yl)-3-hydroxypropyl]-N-pentylpentan-1-aminium pH 5.0, temperature not specified in the publication 708121 3.4.23.39 0.024 - N-[4,4-difluoro-3-oxocyclohexyl]-2-(2-naphthyl)-N-(4-pentylphenyl)-acetamide pH 5.0, 37°C 710185 3.4.23.39 0.0243 - 2-amino-3-[(oxolan-2-yl)methyl]quinazolin-4(3H)-one pH and temperature not specified in the publication 754378 3.4.23.39 0.0244 - (3S,4S)-pyrrolidine-3,4-diyl dibenzoate pH and temperature not specified in the publication 754374 3.4.23.39 0.0305 - 1-(4-nitrophenyl)-2-[2-(pyridin-2-yl)-1H-benzimidazol-1-yl]ethanone pH 5.0, temperature not specified in the publication 717364 3.4.23.39 0.032 - N-[3-(9H-fluoren-2-yl)-3-hydroxypropyl]-N-pentylpentan-1-aminium pH 5.0, temperature not specified in the publication 708121 3.4.23.39 0.038 - (1SR,4RS)-3,3-difluoro-4-hydroxy-N-[2-(2-naphthyl)ethyl]-N(4-pentylphenyl)cyclohexanecarboxamide pH 5.0, 37°C 710185 3.4.23.39 0.0396 - N-[2-(dibutylamino)ethyl]-4-propyl-N-[4-(trifluoromethyl)benzyl]benzamide IC50: 0.0396 mM 668255 3.4.23.39 0.043 - (1RS,4RS)-3,3-difluoro-4-hydroxy-N-[2-(2-naphthyl)ethyl]-N(4-pentylphenyl)cyclohexanecarboxamide pH 5.0, 37°C 710185 3.4.23.39 0.056 - 5-[bis[(benzyloxy)carbonyl]amino]-6-[[1-hydrazinyl-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]amino]-6-oxohexan-1-aminium pH 5.0, temperature not specified in the publication 708121 3.4.23.39 0.062 - 3-[3-(4-chlorophenyl)-3-hydroxy-3-phenylpropyl]-3-azoniabicyclo[4.2.1]nonane pH 5.0, temperature not specified in the publication 708121 3.4.23.39 0.07 - (1S,2S,3R,4R)-2-([4-[3-(1,3-benzodioxol-5-yl)propyl]benzyl]oxy)-3-(naphthalen-2-ylmethoxy)-7-azabicyclo[2.2.1]heptane pH and temperature not specified in the publication 754374 3.4.23.39 0.094 - N-(2,5-dimethyl-1H-pyrrol-1-yl)-4-hydroxybenzamide pH and temperature not specified in the publication 754378 3.4.23.39 0.095 - N,N-dibutyl-3-(1,4-dihydronaphthalen-1-yl)-3-hydroxybutan-1-aminium pH 5.0, temperature not specified in the publication 708121 3.4.23.39 0.1 - N-(3-carbamoylthiophen-2-yl)thiophene-2-carboxamide pH and temperature not specified in the publication 754378 3.4.23.39 0.1 - N-([(1RS)-3,3-difluoro-4-oxocyclopentyl]methyl)-2-(2-naphthyl)-N-(4-pentylphenyl)acetamide value above, pH 5.0, 37°C 710185 3.4.23.39 0.1 - N-([(1SR,4RS)-3,3-difluoro-4-hydroxycyclopentyl]methyl)-2-(2-naphthyl)-N-(4-pentylphenyl)acetamide value above, pH 5.0, 37°C 710185 3.4.23.39 0.1 - N-([(1SR,4SR)-3,3-difluoro-4-hydroxycyclopentyl]methyl)-2-(2-naphthyl)-N-(4-pentylphenyl)acetamide value above, pH 5.0, 37°C 710185 3.4.23.39 0.125 - 1-amino-3-(4-nitroanilino)propan-2-ol pH and temperature not specified in the publication 754378 3.4.23.39 0.15 - (2E)-2-[(2H-1,3-benzodioxol-5-yl)methylidene]hydrazine-1-carboximidamide pH and temperature not specified in the publication 754378 3.4.23.39 0.15 - 4-(imidazo[2,1-b][1,3]thiazol-6-yl)aniline pH and temperature not specified in the publication 754378 3.4.23.39 0.152 - 5-methyl-N3-phenyl-1H-pyrazole-3,4-diamine pH and temperature not specified in the publication 754378 3.4.23.39 0.184 - 4-(1,2-benzothiazol-3-yl)-N-methylpiperazine-1-carboxamide pH and temperature not specified in the publication 754378 3.4.23.39 0.196 - 1-(diphenylmethyl)azetidin-3-ol pH and temperature not specified in the publication 754378 3.4.23.39 0.2 - 1-phenyl-N-(propan-2-yl)methanesulfonamide pH and temperature not specified in the publication 754378 3.4.23.39 0.7 - (1R,2R,3S,4S)-2,3-bis(naphthalen-2-ylmethoxy)-7-azabicyclo[2.2.1]heptane pH and temperature not specified in the publication 754374 3.4.23.39 1 - (1S,2S,3R,4R)-2-[(4-bromobenzyl)oxy]-3-(naphthalen-2-ylmethoxy)-7-azabicyclo[2.2.1]heptane pH and temperature not specified in the publication 754374 3.4.23.39 100 - Lac-Val-Sta-Ala-Sta IC50: 100 mM 648193