3.4.24.82 additional information - additional information Ki(app) of N-terminal alanine-extension mutants and of position [-1] mutants of N-terminal inhibitory domain of tissue inhibitor of metalloproteinases 3 707445 3.4.24.82 0.000003 - (2S,3R)-2-[(cyclopropylmethyl)amino]-N1-hydroxy-N4-[(1S,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]-3-methylbutanediamide or above, pH not specified in the publication, temperature not specified in the publication 734700 3.4.24.82 0.0000033 - tissue inhibitor of matrix metalloproteinases-3 - 668343 3.4.24.82 0.0000079 - TIMP-3 - 680792 3.4.24.82 0.00002 - tinzaparin - 668343 3.4.24.82 0.0000228 - SC81956 at 37°C 678287 3.4.24.82 0.000065 - (2R)-N4-hydroxy-2-(3-hydroxybenzyl)-N1-[(1S,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]butanediamide or above, pH not specified in the publication, temperature not specified in the publication 734700 3.4.24.82 0.000079 - marimastat pH not specified in the publication, temperature not specified in the publication 734700 3.4.24.82 0.00008 - enoxaparin - 668343 3.4.24.82 0.0001 - N-terminal domain of tissue inhibitor of metalloproteinases-3 pH 7.5, 37°C, isoenzyme ADAMTS4-3 709790 3.4.24.82 0.000105 - GGWGPWGPWGDCSRTCGGG - 638958 3.4.24.82 0.00013 - N-terminal domain of tissue inhibitor of metalloproteinases-3 pH 7.5, 37°C, isoenzyme ADAMTS4-1 709790 3.4.24.82 0.00018 - N-terminal domain of tissue inhibitor of metalloproteinases-3 pH 7.5, 37°C, isoenzyme ADAMTS4-2 709790 3.4.24.82 0.00022 - tissue inhibitor of metalloproteinases-3 pH 7.5, 37°C, isoenzyme ADAMTS4-1 709790 3.4.24.82 0.00022 - tissue inhibitor of metalloproteinases-3 pH 7.5, 37°C, isoenzyme ADAMTS4-2 709790 3.4.24.82 0.0004 - tissue inhibitor of metalloproteinases-3 pH 7.5, 37°C, isoenzyme ADAMTS4-3 709790 3.4.24.82 0.00051 - tissue inhibitor of metalloproteinases-3 pH 7.5, 37°C, isoenzyme ADAMTS4-4 709790 3.4.24.82 0.00064 - N-terminal domain of tissue inhibitor of metalloproteinases-3 pH 7.5, 37°C, isoenzyme ADAMTS4-4 709790 3.4.24.82 0.00268 - (E)-4-[2-(3,5-dihydroxyphenyl)ethenyl]1,2-benzenediol pH 7.5, 37°C, substrate: C6-(Gly-Pro-Hyp-Pro-Hyp-Gly)2-Gly-Pro-Hyp-Gly-Thr-Lys(7-methoxycoumarin-4-yl)-Gly-Glu–Leu–Glu–Gly-Arg–Gly-Thr-Lys(Dnp)-Gly-Ile-Ser-(Gly-Pro-Hyp-Pro-Hyp-Gly)2-Gly-Pro-Hyp-NH2 708082 3.4.24.82 0.00506 - (E)-4-[2-(3,5-dihydroxyphenyl)ethenyl]1,2-benzenediol pH 7.5, 37°C, substrate: pH 7.5, 37°C, substrate: Lys(7-methoxycoumarin-4-yl)-Lys-Gln-Glu-Phe-Arg-Gly-Gln-Thr-Lys(Dnp)-NH2 708082 3.4.24.82 0.00634 - pyrogallol pH 7.5, 37°C, substrate: C6-(Gly-Pro-Hyp-Pro-Hyp-Gly)2-Gly-Pro-Hyp-Gly-Thr-Lys(7-methoxycoumarin-4-yl)-Gly-Glu–Leu–Glu–Gly-Arg–Gly-Thr-Lys(Dnp)-Gly-Ile-Ser-(Gly-Pro-Hyp-Pro-Hyp-Gly)2-Gly-Pro-Hyp-NH2 708082 3.4.24.82 0.026 - QEYKAHHSYKLMS at 37°C 678287 3.4.24.82 0.041 - pyrogallol pH 7.5, 37°C, substrate: Lys(7-methoxycoumarin-4-yl)-Lys-Gln-Glu-Phe-Arg-Gly-Gln-Thr-Lys(Dnp)-NH2 708082 3.4.24.82 0.0453 - doxycycline rhADAMTS4(F213-R695), pH and temperature not specified in the publication 709662 3.4.24.82 0.0611 - doxycycline rhADAMTS4(F213-A579), pH and temperature not specified in the publication 709662 3.4.24.82 0.0869 - minocycline rhADAMTS4(F213-R695), pH and temperature not specified in the publication 709662 3.4.24.82 0.0973 - minocycline rhADAMTS4(F213-A579), pH and temperature not specified in the publication 709662 3.4.24.82 0.12 - tetracycline rhADAMTS4(F213-A579), pH and temperature not specified in the publication 709662 3.4.24.82 0.761 - tetracycline rhADAMTS4(F213-R695), pH and temperature not specified in the publication 709662