3.4.22.52 0.00000018 - penetratin pH and temperature not specified in the publication 708257 3.4.22.52 0.00000019 - acetyl-RRMKWKKDPMSSTYIEELGKREVTIPPKYRELLA-NH2 pH and temperature not specified in the publication 708257 3.4.22.52 0.0000002 - acetyl-DPMSSTYIEELGKREVTIPPKYRELLA-NH2 pH and temperature not specified in the publication 708257 3.4.22.52 0.0000005 - acetyl-DPMSSTYIEELGKREVTIPPKYREL-NH2 pH 7.5, 12°C 678542 3.4.22.52 0.0000005 - PCP1B peptide pH and temperature not specified in the publication 708257 3.4.22.52 0.0000006 - acetyl-SSTYIEELGKREVTIPPKYRELLA-NH2 pH 7.5, 12°C 678542 3.4.22.52 0.0000008 - acetyl-DPMSSTYIEELGKREVTIPPKYR-NH2 pH 7.5, 12°C 678542 3.4.22.52 0.0000022 - acetyl-TYIEELGKREVTIPPKYRELLA-NH2 pH 7.5, 12°C 678542 3.4.22.52 0.0000047 - N-[(2S)-4-(2-benzylhydrazinyl)-3,4-dioxo-1-phenylbutan-2-yl]-N2-[(benzyloxy)carbonyl]-L-leucinamide pH and temperature not specified in the publication 708257 3.4.22.52 0.0000085 - 3-([N-[(benzyloxy)carbonyl]-L-leucyl]amino)-2-oxo-4-phenylbutanoic acid pH and temperature not specified in the publication 708257 3.4.22.52 0.000009 - N-(4-amino-3,4-dioxo-1-phenylbutan-2-yl)-1-(1-benzothiophen-2-ylcarbonyl)piperidine-4-carboxamide pH and temperature not specified in the publication 708257 3.4.22.52 0.00002 - N-[1-(4-bromophenyl)-4-(ethylamino)-3,4-dioxobutan-2-yl]-N2-[5-(1,2-dithiolan-3-yl)pentanoyl]-L-leucinamide pH and temperature not specified in the publication 708257 3.4.22.52 0.000026 - acetyl-SSTTYIEELGKREVTIPPKYR-NH2 pH and temperature not specified in the publication 708257 3.4.22.52 0.000026 - acetyl-SSTYIEELGKREVTIPPKYR-NH2 pH 7.5, 12°C 678542 3.4.22.52 0.000026 - CP1B peptide pH and temperature not specified in the publication 707531 3.4.22.52 0.000026 - N-(4-amino-3,4-dioxo-1-phenylbutan-2-yl)-5-oxo-1-[3-(trifluoromethyl)benzyl]-D-prolinamide pH and temperature not specified in the publication 753012 3.4.22.52 0.000027 - N-(4-amino-3,4-dioxo-1-phenylbutan-2-yl)-2-[(E)-2-[4-[(diethylamino)methyl]phenyl]ethenyl]benzamide pH and temperature not specified in the publication 708257 3.4.22.52 0.000036 - N-(4-amino-3,4-dioxo-1-phenylbutan-2-yl)-1-[2-methoxy-6-(trifluoromethyl)benzyl]-5-oxo-D-prolinamide pH and temperature not specified in the publication 753012 3.4.22.52 0.000039 - N-(4-amino-3,4-dioxo-1-phenylbutan-2-yl)-1-benzyl-5-oxo-D-prolinamide pH and temperature not specified in the publication 753012 3.4.22.52 0.000046 - N-(1-amino-1,2-dioxoheptan-3-yl)-1-benzyl-5-oxo-D-prolinamide pH and temperature not specified in the publication 753012 3.4.22.52 0.000048 - 1-benzyl-N-[4-[(4-fluorophenyl)amino]-3,4-dioxo-1-phenylbutan-2-yl]-5-oxo-D-prolinamide pH and temperature not specified in the publication 753012 3.4.22.52 0.00005 - (4S)-N-(4-amino-3,4-dioxo-1-phenylbutan-2-yl)-1-benzyl-4-methyl-5-oxo-D-prolinamide pH and temperature not specified in the publication 753012 3.4.22.52 0.00005 - 4-(4-bromophenyl)-3-([N-[5-(1,2-dithiolan-3-yl)pentanoyl]-L-leucyl]amino)-2-oxobutanoic acid pH and temperature not specified in the publication 708257 3.4.22.52 0.00005 - N-[4-(cyclopropylamino)-3,4-dioxo-1-phenylbutan-2-yl]-5-oxo-1-[2-(trifluoromethoxy)benzyl]-D-prolinamide pH and temperature not specified in the publication 753012 3.4.22.52 0.000057 - N-(4-amino-3,4-dioxo-1-phenylbutan-2-yl)-5-oxo-1-[2-(trifluoromethoxy)benzyl]-D-prolinamide pH and temperature not specified in the publication 753012 3.4.22.52 0.000059 - N-(4-amino-3,4-dioxo-1-phenylbutan-2-yl)-5-oxo-1-[2-(trifluoromethyl)benzyl]-D-prolinamide pH and temperature not specified in the publication 753012 3.4.22.52 0.000064 - (2R)-N-(4-amino-3,4-dioxo-1-phenylbutan-2-yl)-1-benzyl-6-oxopiperidine-2-carboxamide pH and temperature not specified in the publication 753012 3.4.22.52 0.00007 - 1-benzyl-N-[3,4-dioxo-1-phenyl-4-(phenylamino)butan-2-yl]-5-oxo-D-prolinamide pH and temperature not specified in the publication 753012 3.4.22.52 0.000073 - 1-(2-chlorobenzyl)-N-[4-(cyclopropylamino)-3,4-dioxo-1-phenylbutan-2-yl]-5-oxo-D-prolinamide pH and temperature not specified in the publication 753012 3.4.22.52 0.000081 - 1-[(4-methylphenyl)sulfonyl]-N-(1-oxo-3-phenylpropan-2-yl)-D-prolinamide pH and temperature not specified in the publication 708257 3.4.22.52 0.000082 - N-(4-amino-3,4-dioxo-1-phenylbutan-2-yl)-1-benzyl-6-oxo-1,6-dihydropyridine-2-carboxamide pH and temperature not specified in the publication 753012 3.4.22.52 0.00009 - N-[4-(cyclopropylamino)-3,4-dioxo-1-phenylbutan-2-yl]-5-oxo-1-[2-(trifluoromethyl)benzyl]-D-prolinamide pH and temperature not specified in the publication 753012 3.4.22.52 0.000093 - acetyl-TYIEELGKREVTIPPKYR-NH2 pH 7.5, 12°C 678542 3.4.22.52 0.000093 - acetyl-TYIEELGKREVTIPPKYR-NH2 pH and temperature not specified in the publication 708257 3.4.22.52 0.000101 - (4R)-N-(4-amino-3,4-dioxo-1-phenylbutan-2-yl)-3-benzyl-1-methyl-2-oxoimidazolidine-4-carboxamide pH and temperature not specified in the publication 753012 3.4.22.52 0.00011 - 1-benzyl-N-[4-(cyclobutylamino)-3,4-dioxo-1-phenylbutan-2-yl]-5-oxo-D-prolinamide pH and temperature not specified in the publication 753012 3.4.22.52 0.000125 - N-(4-amino-3,4-dioxo-1-phenylbutan-2-yl)-5-oxo-1-[3-(trifluoromethoxy)benzyl]-D-prolinamide pH and temperature not specified in the publication 753012 3.4.22.52 0.000129 - N-(4-amino-3,4-dioxo-1-phenylbutan-2-yl)-1-[(4-methylphenyl)sulfonyl]-D-prolinamide pH and temperature not specified in the publication 753012 3.4.22.52 0.00013 - 1-benzyl-N-[4-(cyclopropylamino)-3,4-dioxo-1-phenylbutan-2-yl]-5-oxo-D-prolinamide pH and temperature not specified in the publication 753012 3.4.22.52 0.000165 - 1-benzyl-N-[4-(ethylamino)-3,4-dioxo-1-phenylbutan-2-yl]-5-oxo-D-prolinamide pH and temperature not specified in the publication 753012 3.4.22.52 0.00018 - N-(4-amino-3,4-dioxo-1-phenylbutan-2-yl)-5-oxo-1-(pyridin-4-ylmethyl)-D-prolinamide pH and temperature not specified in the publication 753012 3.4.22.52 0.0002 - N2-[(benzyloxy)carbonyl]-N-[4-(ethylamino)-3,4-dioxo-1-phenylbutan-2-yl]-L-leucinamide pH and temperature not specified in the publication 708257 3.4.22.52 0.00024 - N-[4-(cyclopropylamino)-3,4-dioxo-1-phenylbutan-2-yl]-5-oxo-1-[2-(trifluoromethoxy)-6-(trifluoromethyl)benzyl]-D-prolinamide pH and temperature not specified in the publication 753012 3.4.22.52 0.000268 - N-(4-amino-3,4-dioxo-1-phenylbutan-2-yl)-1-(cyclohexylmethyl)-5-oxo-D-prolinamide pH and temperature not specified in the publication 753012 3.4.22.52 0.000268 - N-(4-amino-3,4-dioxo-1-phenylbutan-2-yl)-2-benzyl-1,2-thiazolidine-3-carboxamide 1,1-dioxide pH and temperature not specified in the publication 753012 3.4.22.52 0.000528 - N-(4-amino-3,4-dioxo-1-phenylbutan-2-yl)-1-benzyl-5-oxo-L-prolinamide pH and temperature not specified in the publication 753012 3.4.22.52 0.00053 - N-[4-(cyclopropylamino)-3,4-dioxo-1-phenylbutan-2-yl]-1-(1-methyl-1H-pyrazol-4-yl)-5-oxo-D-prolinamide pH and temperature not specified in the publication 753012 3.4.22.52 0.000545 - N-[4-(cyclopropylamino)-3,4-dioxo-1-phenylbutan-2-yl]-1-(2,3-dihydro-1H-inden-2-yl)-5-oxo-D-prolinamide pH and temperature not specified in the publication 753012 3.4.22.52 0.00097 - N-[4-(cyclopropylamino)-3,4-dioxo-1-phenylbutan-2-yl]-5-oxo-D-prolinamide pH and temperature not specified in the publication 753012 3.4.22.52 0.00135 - N-(4-amino-3,4-dioxo-1-phenylbutan-2-yl)-1-(2,2-dimethylpropyl)-5-oxo-D-prolinamide pH and temperature not specified in the publication 753012 3.4.22.52 0.0018 - ethyl 3-([N-[(benzyloxy)carbonyl]-L-leucyl]amino)-2-oxo-4-phenylbutanoate pH and temperature not specified in the publication 708257 3.4.22.52 0.0024 - acetyl-DPMSSTYIEELGKREVT-betaAla-PPKYRELLA-NH2 pH and temperature not specified in the publication 708257 3.4.22.52 0.00436 - 1-benzyl-N-[4-(methoxyamino)-3,4-dioxo-1-phenylbutan-2-yl]-5-oxo-D-prolinamide pH and temperature not specified in the publication 753012 3.4.22.52 0.0059 - ritonavir - 644006 3.4.22.52 0.0069 - acetyl-DPMSSTYIEELGK-NH2 pH 7.5, 12°C 678542 3.4.22.52 0.01 - ethyl 4-(4-bromophenyl)-3-([N-[5-(1,2-dithiolan-3-yl)pentanoyl]-L-leucyl]amino)-2-oxobutanoate IC50 above 0.01 mM, pH and temperature not specified in the publication 708257 3.4.22.52 0.0117 - acetyl-SSTYIEELGK-NH-(CH2O)2-CH2C(O)-TIPPKYR-NH2 pH 7.5, 12°C 678542 3.4.22.52 0.017 - acetyl-DPMSSTYIEE-betaAla-GKREVTIPPKYRELLA-NH2 pH and temperature not specified in the publication 708257 3.4.22.52 0.017 - acetyl-SSTYIEELGKREVTIPPK-NH2 pH 7.5, 12°C 678542 3.4.22.52 0.035 - acetyl-REVTIPPKYRELLA-NH2 pH 7.5, 12°C 678542 3.4.22.52 0.726 - acetyl-RYKPPITVERKGLEEIYTSS-NH2 pH 7.5, 12°C 678542