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Literature summary extracted from

  • Oliva, M.L.V.; Andrade, S.; Batista, I.F.C.; Sampaio, M.U.; Juliano, M.; Fritz, H.; Auerswald, E.A.; Sampaio, C.A.M.
    Human plasma kallikrein and tissue kallikrein binding to a substrate based on the reactive site of a factor Xa inhibitor isolates from Bauhinia ungulata seeds (1999), Immunopharmacology, 45, 145-149.
    View publication on PubMed

Inhibitors

EC Number Inhibitors Comment Organism Structure
3.4.21.34 Bauhinia unglata factor Xa inhibitor
-
Homo sapiens
3.4.21.34 Soybean trypsin inhibitor
-
Homo sapiens
3.4.21.35 additional information no inhibition by Bauhinia ungulata factor Xa inhibitor, and Bauhinia variegata trypsin inhibitor Sus scrofa
3.4.21.35 Soybean trypsin inhibitor no inhibition Sus scrofa

KM Value [mM]

EC Number KM Value [mM] KM Value Maximum [mM] Substrate Comment Organism Structure
3.4.21.35 additional information
-
additional information
-
Sus scrofa
3.4.21.35 0.00023
-
o-aminobenzoyl-VMIAALPRTMFIQ-N-(2,4-dinitrophenyl)ethylene diamine pH 8.0, 37°C Sus scrofa
3.4.21.35 0.0005
-
o-aminobenzoyl-VMIAALPRTMQ-N-(2,4-dinitrophenyl)ethylene diamine pH 8.0, 37°C Sus scrofa
3.4.21.35 0.0007
-
o-aminobenzoyl-LPRTMQ-N-(2,4-dinitrophenyl)ethylene diamine pH 8.0, 37°C Sus scrofa
3.4.21.35 0.0027
-
o-aminobenzoyl-LPRTMFIQ-N-(2,4-dinitrophenyl)ethylene diamine pH 8.0, 37°C Sus scrofa

Natural Substrates/ Products (Substrates)

EC Number Natural Substrates Organism Comment (Nat. Sub.) Natural Products Comment (Nat. Pro.) Rev. Reac.
3.4.21.35 polypeptide + H2O Sus scrofa
-
peptides
-
?

Organism

EC Number Organism UniProt Comment Textmining
3.4.21.34 Homo sapiens
-
-
-
3.4.21.34 Sus scrofa
-
-
-
3.4.21.35 Sus scrofa
-
-
-

Source Tissue

EC Number Source Tissue Comment Organism Textmining
3.4.21.34 pancreas
-
Sus scrofa
-
3.4.21.34 plasma
-
Homo sapiens
-
3.4.21.34 plasma
-
Sus scrofa
-
3.4.21.35 pancreas
-
Sus scrofa
-

Substrates and Products (Substrate)

EC Number Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
3.4.21.34 additional information based on the reactive site sequence of Bauhinia ungulata Xa inhibitor peptides Homo sapiens ?
-
?
3.4.21.34 additional information based on the reactive site sequence of Bauhinia ungulata Xa inhibitor peptides Sus scrofa ?
-
?
3.4.21.35 o-aminobenzoyl-LPRTMFIQ-N-(2,4-dinitrophenyl)ethylene diamine + H2O shortened, quenched fluorescent substrate, synthesized based on Bauhinia ungulata factor Xa inhibitor reactive sequence site Sus scrofa ?
-
?
3.4.21.35 o-aminobenzoyl-LPRTMQ-N-(2,4-dinitrophenyl)ethylene diamine + H2O shortened, quenched fluorescent substrate, synthesized based on Bauhinia ungulata factor Xa inhibitor reactive sequence site Sus scrofa ?
-
?
3.4.21.35 o-aminobenzoyl-VMIAALPRTMFIQ-N-(2,4-dinitrophenyl)ethylene diamine + H2O low activity Sus scrofa ?
-
?
3.4.21.35 o-aminobenzoyl-VMIAALPRTMFIQ-N-(2,4-dinitrophenyl)ethylene diamine + H2O quenched fluorescent substrate, synthesized based on Bauhinia ungulata factor Xa inhibitor reactive sequence site Sus scrofa ?
-
?
3.4.21.35 o-aminobenzoyl-VMIAALPRTMQ-N-(2,4-dinitrophenyl)ethylene diamine + H2O low activity Sus scrofa ?
-
?
3.4.21.35 o-aminobenzoyl-VMIAALPRTMQ-N-(2,4-dinitrophenyl)ethylene diamine + H2O quenched fluorescent substrate, synthesized based on Bauhinia ungulata factor Xa inhibitor reactive sequence site Sus scrofa ?
-
?
3.4.21.35 polypeptide + H2O
-
Sus scrofa peptides
-
?

Temperature Optimum [°C]

EC Number Temperature Optimum [°C] Temperature Optimum Maximum [°C] Comment Organism
3.4.21.34 37
-
assay at Homo sapiens
3.4.21.34 37
-
assay at Sus scrofa
3.4.21.35 37
-
assay at Sus scrofa

Turnover Number [1/s]

EC Number Turnover Number Minimum [1/s] Turnover Number Maximum [1/s] Substrate Comment Organism Structure
3.4.21.35 additional information
-
additional information
-
Sus scrofa
3.4.21.35 0.0005
-
o-aminobenzoyl-VMIAALPRTMFIQ-N-(2,4-dinitrophenyl)ethylene diamine pH 8.0, 37°C Sus scrofa
3.4.21.35 0.004
-
o-aminobenzoyl-VMIAALPRTMQ-N-(2,4-dinitrophenyl)ethylene diamine pH 8.0, 37°C Sus scrofa
3.4.21.35 0.014
-
o-aminobenzoyl-LPRTMQ-N-(2,4-dinitrophenyl)ethylene diamine pH 8.0, 37°C Sus scrofa
3.4.21.35 0.032
-
o-aminobenzoyl-LPRTMFIQ-N-(2,4-dinitrophenyl)ethylene diamine pH 8.0, 37°C Sus scrofa

pH Optimum

EC Number pH Optimum Minimum pH Optimum Maximum Comment Organism
3.4.21.35 8
-
assay at Sus scrofa