EC Number | Inhibitors | Comment | Organism | Structure |
---|---|---|---|---|
3.4.14.2 | bestatin | 1 mM, 12% inhibition of DPP II-S, 21% inhibition of DPP II-M; no inhibition | Rattus norvegicus | |
3.4.14.2 | diisopropyl fluorophosphate | - |
Rattus norvegicus | |
3.4.14.2 | additional information | no inhibition by bacitracin | Rattus norvegicus | |
3.4.14.2 | N6-benzyloxycarbonyl-Lys-Pro | 1 mM, 31% inhibition of DPP II-S, 41% inhibition of DPP II-M | Rattus norvegicus | |
3.4.14.2 | Na+ | 400 mM NaCl, 56% inhibition of DPP II-M, 31% inhibition of DPP II-S | Rattus norvegicus | |
3.4.14.2 | p-hydroxymercuribenzoate | - |
Rattus norvegicus | |
3.4.14.2 | phenylmethylsulfonyl fluoride | - |
Rattus norvegicus | |
3.4.14.2 | Tris | - |
Rattus norvegicus |
EC Number | KM Value [mM] | KM Value Maximum [mM] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|---|
3.4.14.2 | 0.018 | - |
Gly-Pro-4-nitroanilide | enzyme form DPP II-S | Rattus norvegicus | |
3.4.14.2 | 0.032 | - |
Gly-Pro-4-nitroanilide | enzyme form DPP II-M | Rattus norvegicus | |
3.4.14.2 | 0.068 | - |
Arg-Pro-4-nitroanilide | enzyme form DPP II-M | Rattus norvegicus | |
3.4.14.2 | 0.087 | - |
Lys-Ala-2-naphthylamide | enzyme form DPP II-S | Rattus norvegicus | |
3.4.14.2 | 0.21 | - |
Lys-Ala-2-naphthylamide | enzyme form DPP II-M | Rattus norvegicus | |
3.4.14.2 | 0.502 | - |
His-Pro-Val | enzyme form DPP II-S | Rattus norvegicus |
EC Number | Localization | Comment | Organism | GeneOntology No. | Textmining |
---|---|---|---|---|---|
3.4.14.2 | membrane | enzyme form DPP II-S | Rattus norvegicus | 16020 | - |
3.4.14.2 | soluble | enzyme form DPP II-M | Rattus norvegicus | - |
- |
EC Number | Molecular Weight [Da] | Molecular Weight Maximum [Da] | Comment | Organism |
---|---|---|---|---|
3.4.14.2 | 52500 | - |
2 * 52500, SDS-PAGE | Rattus norvegicus |
3.4.14.2 | 110000 | - |
gel filtration | Rattus norvegicus |
EC Number | Organism | UniProt | Comment | Textmining |
---|---|---|---|---|
3.4.14.2 | Rattus norvegicus | - |
two enzyme forms: DPP II-M and DPP II-S | - |
EC Number | Purification (Comment) | Organism |
---|---|---|
3.4.14.2 | enzyme form DPP II-S and DPP II-M | Rattus norvegicus |
EC Number | Source Tissue | Comment | Organism | Textmining |
---|---|---|---|---|
3.4.14.2 | brain | - |
Rattus norvegicus | - |
3.4.14.2 | hypophysis | - |
Rattus norvegicus | - |
EC Number | Storage Stability | Organism |
---|---|---|
3.4.14.2 | -20°C, pH 6.0, 20 mM BisTris-HCl buffer, stable | Rattus norvegicus |
EC Number | Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|---|
3.4.14.2 | Ala-Ala-2-naphthylamide + H2O | - |
Rattus norvegicus | Ala-Ala + 2-naphthylamine | - |
? | |
3.4.14.2 | Arg-Pro-4-nitroanilide + H2O | - |
Rattus norvegicus | Arg-Pro + 4-nitroaniline | - |
? | |
3.4.14.2 | bradykinin fragment 1-3 + H2O | - |
Rattus norvegicus | ? | - |
? | |
3.4.14.2 | bradykinin fragment 1-5 + H2O | - |
Rattus norvegicus | ? | - |
? | |
3.4.14.2 | Gly-Pro-4-nitroanilide + H2O | - |
Rattus norvegicus | Gly-Pro + 4-nitroaniline | - |
? | |
3.4.14.2 | His-Pro-Val + H2O | - |
Rattus norvegicus | His-Pro + Val | - |
? | |
3.4.14.2 | Lys-Ala-2-naphthylamide + H2O | - |
Rattus norvegicus | Lys-Ala + 2-naphthylamine | - |
? | |
3.4.14.2 | additional information | no activity with bradykinin | Rattus norvegicus | ? | - |
? | |
3.4.14.2 | Phe-Pro-2-naphthylamide + H2O | - |
Rattus norvegicus | Phe-Pro + 2-naphthylamine | - |
? |
EC Number | Subunits | Comment | Organism |
---|---|---|---|
3.4.14.2 | dimer | 2 * 52500, SDS-PAGE | Rattus norvegicus |
EC Number | Synonyms | Comment | Organism |
---|---|---|---|
3.4.14.2 | DPP II | - |
Rattus norvegicus |
EC Number | pH Optimum Minimum | pH Optimum Maximum | Comment | Organism |
---|---|---|---|---|
3.4.14.2 | 5.5 | - |
hydrolysis of Gly-Pro-4-nitroanilide or Arg-Pro-4-nitroanilide | Rattus norvegicus |
EC Number | pH Stability | pH Stability Maximum | Comment | Organism |
---|---|---|---|---|
3.4.14.2 | 3 | - |
4°C, 24 h, loss of activity of DPP II-M | Rattus norvegicus |
3.4.14.2 | 4 | 8 | 4°C, 24 h, DPP II-M is stable | Rattus norvegicus |