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Literature summary extracted from

  • Severson, D.L.; Denton, R.M.; Pask, H.T.; Randle, P.J.
    Calcium and magnesium ions as effectors of adipose-tissue pyruvate dehydrogenase phosphate phosphatase (1974), Biochem. J., 140, 225-237.
    View publication on PubMedView publication on EuropePMC

Inhibitors

EC Number Inhibitors Comment Organism Structure
3.1.3.43 A23187
-
Rattus norvegicus
3.1.3.43 Ni2+
-
Rattus norvegicus
3.1.3.43 ruthenium red
-
Rattus norvegicus

KM Value [mM]

EC Number KM Value [mM] KM Value Maximum [mM] Substrate Comment Organism Structure
3.1.3.43 0.003
-
[Pyruvate dehydrogenase (lipoamide)]-phosphate with Ca2+ and Mg2+ Rattus norvegicus

Localization

EC Number Localization Comment Organism GeneOntology No. Textmining
3.1.3.43 mitochondrion
-
Rattus norvegicus 5739
-
3.1.3.43 mitochondrion
-
Sus scrofa 5739
-

Metals/Ions

EC Number Metals/Ions Comment Organism Structure
3.1.3.43 Ca2+
-
Sus scrofa
3.1.3.43 Ca2+ Km: 0.001 Rattus norvegicus
3.1.3.43 Mg2+
-
Sus scrofa
3.1.3.43 Mg2+ Km: 0.52 mM Rattus norvegicus
3.1.3.43 Sr2+
-
Rattus norvegicus

Natural Substrates/ Products (Substrates)

EC Number Natural Substrates Organism Comment (Nat. Sub.) Natural Products Comment (Nat. Pro.) Rev. Reac.
3.1.3.43 [pyruvate dehydrogenase (lipoamide)]-phosphate + H2O Rattus norvegicus
-
?
-
?
3.1.3.43 [pyruvate dehydrogenase (lipoamide)]-phosphate + H2O Sus scrofa
-
?
-
?

Organism

EC Number Organism UniProt Comment Textmining
3.1.3.43 Rattus norvegicus
-
-
-
3.1.3.43 Sus scrofa
-
-
-

Purification (Commentary)

EC Number Purification (Comment) Organism
3.1.3.43 partially Sus scrofa

Source Tissue

EC Number Source Tissue Comment Organism Textmining
3.1.3.43 adipose
-
Rattus norvegicus
-
3.1.3.43 epididymis
-
Rattus norvegicus
-
3.1.3.43 heart
-
Rattus norvegicus
-
3.1.3.43 heart
-
Sus scrofa
-

Substrates and Products (Substrate)

EC Number Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
3.1.3.43 [pyruvate dehydrogenase (lipoamide)]-phosphate + H2O
-
Rattus norvegicus [pyruvate dehydrogenase (lipoamide)] + phosphate
-
ir
3.1.3.43 [pyruvate dehydrogenase (lipoamide)]-phosphate + H2O
-
Sus scrofa [pyruvate dehydrogenase (lipoamide)] + phosphate
-
ir
3.1.3.43 [pyruvate dehydrogenase (lipoamide)]-phosphate + H2O
-
Rattus norvegicus ?
-
?
3.1.3.43 [pyruvate dehydrogenase (lipoamide)]-phosphate + H2O
-
Sus scrofa ?
-
?