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Literature summary extracted from

  • Seward, H.E.; Roujeinikova, A.; McLean, K.J.; Munro, A.W.; Leys, D.
    Crystal structure of the Mycobacterium tuberculosis P450 CYP121-fluconazole complex reveals new azole drug-P450 binding mode (2006), J. Biol. Chem., 281, 39437-39443.
    View publication on PubMed

Cloned(Commentary)

EC Number Cloned (Comment) Organism
1.14.19.70
-
Mycobacterium tuberculosis

Crystallization (Commentary)

EC Number Crystallization (Comment) Organism
1.14.19.70 fluconazole-bound CYP121, sitting drop vapor diffusion method, using 20% (w/v) polyethylene glycol 3350 and 0.2 M NaSCN Mycobacterium tuberculosis

Inhibitors

EC Number Inhibitors Comment Organism Structure
1.14.19.70 fluconazole
-
Mycobacterium tuberculosis

Organism

EC Number Organism UniProt Comment Textmining
1.14.19.70 Mycobacterium tuberculosis P9WPP7
-
-
1.14.19.70 Mycobacterium tuberculosis H37Rv P9WPP7
-
-

Purification (Commentary)

EC Number Purification (Comment) Organism
1.14.19.70
-
Mycobacterium tuberculosis

Subunits

EC Number Subunits Comment Organism
1.14.19.70 homohexamer x-ray crystallography Mycobacterium tuberculosis

Synonyms

EC Number Synonyms Comment Organism
1.14.19.70 CYP121
-
Mycobacterium tuberculosis

Cofactor

EC Number Cofactor Comment Organism Structure
1.14.19.70 heme
-
Mycobacterium tuberculosis