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Literature summary extracted from

  • Font, M.; Dominguez, M.J.; Sanmartin, C.; Palop, J.A.; San-Francisco, S.; Urrutia, O.; Houdusse, F.; Garcia-Mina, J.M.
    Structural characteristics of phosphoramide derivatives as urease inhibitors. Requirements for activity (2008), J. Agric. Food Chem., 56, 8451-8460.
    View publication on PubMed

Inhibitors

EC Number Inhibitors Comment Organism Structure
3.5.1.5 3,5-dimethylphenyl diamidophosphate
-
 Canavalia ensiformis
3.5.1.5 4-(benzyloxy)phenyl diamidophosphate
-
 Canavalia ensiformis
3.5.1.5 4-nitrophenyl diamidophosphate
-
 Canavalia ensiformis
3.5.1.5 N-(2-methoxy-4-nitrophenyl)phosphoric triamide
-
 Canavalia ensiformis
3.5.1.5 N-(2-nitrophenyl)phosphoric triamide
-
 Canavalia ensiformis
3.5.1.5 N-(2-phenylethyl)phosphoric triamide
-
 Canavalia ensiformis
3.5.1.5 N-(2-phenylethyl)phosphorothioic triamide
-
 Canavalia ensiformis
3.5.1.5 N-(3-methoxyphenyl)phosphoric triamide
-
 Canavalia ensiformis
3.5.1.5 N-(3-methylpyridin-2-yl)phosphorothioic triamide
-
 Canavalia ensiformis
3.5.1.5 N-(3-morpholin-2-ylpropyl)phosphoric triamide
-
 Canavalia ensiformis
3.5.1.5 N-(3-nitropyridin-2-yl)phosphoric triamide
-
 Canavalia ensiformis
3.5.1.5 N-(4-cyclohexylphenyl)phosphoric triamide
-
 Canavalia ensiformis
3.5.1.5 N-(4-methoxy-1,3-benzothiazol-2-yl)phosphoric triamide
-
 Canavalia ensiformis
3.5.1.5 N-(4-methyl-1,3-benzothiazol-2-yl)phosphoric triamide
-
 Canavalia ensiformis
3.5.1.5 N-(4-methyl-2-nitrophenyl)phosphoric triamide
-
 Canavalia ensiformis
3.5.1.5 N-(4-nitrophenyl)phosphoric triamide
-
 Canavalia ensiformis
3.5.1.5 N-(4-phenoxyphenyl)phosphoric triamide
-
 Canavalia ensiformis
3.5.1.5 N-(6-ethoxy-1,3-benzothiazol-2-yl)phosphoric triamide
-
 Canavalia ensiformis
3.5.1.5 N-(6-fluoro-1,3-benzothiazol-2-yl)phosphoric triamide
-
 Canavalia ensiformis
3.5.1.5 N-1,3-benzothiazol-2-ylphosphoric triamide
-
 Canavalia ensiformis
3.5.1.5 N-1,3-benzothiazol-2-ylphosphorothioic triamide
-
 Canavalia ensiformis
3.5.1.5 N-adamant-1-ylphosphoric triamide
-
 Canavalia ensiformis
3.5.1.5 N-n-butylphosphoric triamide
-
 Canavalia ensiformis
3.5.1.5 N-n-butylthiophosphoric triamide
-
 Canavalia ensiformis
3.5.1.5 N-naphthalen-1-ylphosphoric triamide
-
 Canavalia ensiformis
3.5.1.5 N-phenylphosphoric triamide
-
 Canavalia ensiformis
3.5.1.5 N-[2-(4-fluorophenyl)ethyl]phosphoric triamide
-
 Canavalia ensiformis
3.5.1.5 N-[2-(difluoromethoxy)phenyl]phosphoric triamide
-
 Canavalia ensiformis
3.5.1.5 N-[2-(trifluoromethoxy)phenyl]phosphoric triamide
-
 Canavalia ensiformis
3.5.1.5 N-[4-(benzyloxy)phenyl]phosphoric triamide
-
 Canavalia ensiformis
3.5.1.5 O-[4-(benzyloxy)phenyl] diamidothiophosphate
-
 Canavalia ensiformis
3.5.1.5 phenylphosphorodiamidate
-
 Canavalia ensiformis

Organism

EC Number Organism UniProt Comment Textmining
3.5.1.5 Canavalia ensiformis
-
 Jack bean
-

Substrates and Products (Substrate)

EC Number Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
3.5.1.5 urea + H2O
-
 Canavalia ensiformis CO2 + 2 NH3
-
 ?

Synonyms

EC Number Synonyms Comment Organism
3.5.1.5 urease
-
 Canavalia ensiformis

IC50 Value

EC Number IC50 Value IC50 Value Maximum Comment Organism Inhibitor Structure
3.5.1.5 0.000002
-
-
 Canavalia ensiformis N-1,3-benzothiazol-2-ylphosphoric triamide
3.5.1.5 0.000003
-
-
 Canavalia ensiformis phenylphosphorodiamidate
3.5.1.5 0.000003
-
-
 Canavalia ensiformis N-(4-methyl-2-nitrophenyl)phosphoric triamide
3.5.1.5 0.000005
-
-
 Canavalia ensiformis N-(6-ethoxy-1,3-benzothiazol-2-yl)phosphoric triamide
3.5.1.5 0.000005
-
-
 Canavalia ensiformis N-(6-fluoro-1,3-benzothiazol-2-yl)phosphoric triamide
3.5.1.5 0.00001
-
-
 Canavalia ensiformis N-(4-methoxy-1,3-benzothiazol-2-yl)phosphoric triamide
3.5.1.5 0.00001
-
-
 Canavalia ensiformis N-(4-methyl-1,3-benzothiazol-2-yl)phosphoric triamide
3.5.1.5 0.000014
-
-
 Canavalia ensiformis N-(2-phenylethyl)phosphoric triamide
3.5.1.5 0.000016
-
-
 Canavalia ensiformis 4-(benzyloxy)phenyl diamidophosphate
3.5.1.5 0.00002
-
-
 Canavalia ensiformis N-(2-methoxy-4-nitrophenyl)phosphoric triamide
3.5.1.5 0.00002
-
-
 Canavalia ensiformis N-[2-(difluoromethoxy)phenyl]phosphoric triamide
3.5.1.5 0.000025
-
-
 Canavalia ensiformis 3,5-dimethylphenyl diamidophosphate
3.5.1.5 0.000048
-
-
 Canavalia ensiformis N-[2-(4-fluorophenyl)ethyl]phosphoric triamide
3.5.1.5 0.000063
-
-
 Canavalia ensiformis 4-nitrophenyl diamidophosphate
3.5.1.5 0.00007
-
-
 Canavalia ensiformis N-(3-nitropyridin-2-yl)phosphoric triamide
3.5.1.5 0.0001
-
-
 Canavalia ensiformis N-n-butylthiophosphorictriamide
3.5.1.5 0.0003
-
-
 Canavalia ensiformis N-(4-nitrophenyl)phosphoric triamide
3.5.1.5 0.00053
-
-
 Canavalia ensiformis N-naphthalen-1-ylphosphoric triamide
3.5.1.5 0.00071
-
-
 Canavalia ensiformis N-(3-morpholin-2-ylpropyl)phosphoric triamide
3.5.1.5 0.00256
-
-
 Canavalia ensiformis N-adamant-1-ylphosphoric triamide
3.5.1.5 0.00296
-
-
 Canavalia ensiformis N-1,3-benzothiazol-2-ylphosphorothioic triamide
3.5.1.5 0.003
-
-
 Canavalia ensiformis N-(2-nitrophenyl)phosphoric triamide
3.5.1.5 0.0035
-
-
 Canavalia ensiformis N-[4-(benzyloxy)phenyl]phosphoric triamide
3.5.1.5 0.00363
-
-
 Canavalia ensiformis N-phenylphosphoric triamide
3.5.1.5 0.00557
-
-
 Canavalia ensiformis N-(3-methoxyphenyl)phosphoric triamide
3.5.1.5 0.01298
-
-
 Canavalia ensiformis N-(4-phenoxyphenyl)phosphoric triamide
3.5.1.5 0.01386
-
-
 Canavalia ensiformis N-(2-phenylethyl)phosphorothioic triamide
3.5.1.5 0.01654
-
-
 Canavalia ensiformis O-[4-(benzyloxy)phenyl] diamidothiophosphate
3.5.1.5 0.04255
-
-
 Canavalia ensiformis N-(3-methylpyridin-2-yl)phosphorothioic triamide
3.5.1.5 0.04425
-
-
 Canavalia ensiformis N-(4-cyclohexylphenyl)phosphoric triamide
3.5.1.5 0.075
-
-
 Canavalia ensiformis N-[2-(trifluoromethoxy)phenyl]phosphoric triamide