EC Number | Inhibitors | Comment | Organism | Structure |
---|---|---|---|---|
3.4.24.86 | (3S)-1-[[4-(but-2-yn-1-yloxy)phenyl]sulfonyl]pyrrolidine-3-thiol | - |
Sus scrofa | |
3.4.24.86 | 2-[[4-(but-2-yn-1-ylamino)phenyl]sulfonyl]ethanethiol | - |
Sus scrofa | |
3.4.24.86 | 2-[[4-(but-2-yn-1-yloxy)phenyl]sulfonyl]ethanethiol | - |
Sus scrofa | |
3.4.24.86 | 2-[[[4-(but-2-yn-1-yloxy)phenyl]sulfonyl](methyl)amino]-N-hydroxyacetamide | - |
Sus scrofa | |
3.4.24.86 | 3-[[4-(but-2-yn-1-ylamino)phenyl]sulfonyl]cyclohexanethiol | - |
Sus scrofa | |
3.4.24.86 | 3-[[4-(but-2-yn-1-ylamino)phenyl]sulfonyl]propane-1-thiol | - |
Sus scrofa | |
3.4.24.86 | 3-[[4-(but-2-yn-1-yloxy)phenyl]sulfonyl]cyclohexanethiol | - |
Sus scrofa | |
3.4.24.86 | 3-[[4-(but-2-yn-1-yloxy)phenyl]sulfonyl]cyclopentanethiol | - |
Sus scrofa | |
3.4.24.86 | 3-[[4-(but-2-yn-1-yloxy)phenyl]sulfonyl]propane-1-thiol | - |
Sus scrofa |
EC Number | Organism | UniProt | Comment | Textmining |
---|---|---|---|---|
3.4.24.86 | Sus scrofa | - |
- |
- |
EC Number | Synonyms | Comment | Organism |
---|---|---|---|
3.4.24.86 | TACE | - |
Sus scrofa |
3.4.24.86 | tumor necrosis factor alpha-converting enzyme | - |
Sus scrofa |
EC Number | Ki Value [mM] | Ki Value maximum [mM] | Inhibitor | Comment | Organism | Structure |
---|---|---|---|---|---|---|
3.4.24.86 | 0.000002 | - |
2-[[4-(but-2-yn-1-ylamino)phenyl]sulfonyl]ethanethiol | - |
Sus scrofa | |
3.4.24.86 | 0.0000045 | - |
3-[[4-(but-2-yn-1-ylamino)phenyl]sulfonyl]propane-1-thiol | - |
Sus scrofa | |
3.4.24.86 | 0.000008 | - |
2-[[4-(but-2-yn-1-yloxy)phenyl]sulfonyl]ethanethiol | - |
Sus scrofa | |
3.4.24.86 | 0.00001 | - |
2-[[[4-(but-2-yn-1-yloxy)phenyl]sulfonyl](methyl)amino]-N-hydroxyacetamide | - |
Sus scrofa | |
3.4.24.86 | 0.00001 | - |
3-[[4-(but-2-yn-1-yloxy)phenyl]sulfonyl]propane-1-thiol | - |
Sus scrofa | |
3.4.24.86 | 0.000017 | - |
3-[[4-(but-2-yn-1-ylamino)phenyl]sulfonyl]cyclohexanethiol | - |
Sus scrofa | |
3.4.24.86 | 0.000028 | - |
(3S)-1-[[4-(but-2-yn-1-yloxy)phenyl]sulfonyl]pyrrolidine-3-thiol | - |
Sus scrofa | |
3.4.24.86 | 0.00003 | - |
3-[[4-(but-2-yn-1-yloxy)phenyl]sulfonyl]cyclohexanethiol | - |
Sus scrofa | |
3.4.24.86 | 0.00005 | - |
3-[[4-(but-2-yn-1-yloxy)phenyl]sulfonyl]cyclopentanethiol | - |
Sus scrofa |