EC Number | Inhibitors | Comment | Organism | Structure |
---|---|---|---|---|
3.4.21.26 | (2R)-1-(1-[[3-(azepan-1-ylcarbonyl)phenyl]carbonyl]-L-prolyl)pyrrolidine-2-carbonitrile | 50% inhibition at 4.6 nM | Sus scrofa | |
3.4.21.26 | (2R)-1-(1-[[4-(pyrrolidin-1-ylcarbonyl)phenyl]carbonyl]-L-prolyl)pyrrolidine-2-carbonitrile | 50% inhibition at 1.6 nM | Sus scrofa | |
3.4.21.26 | (2R)-1-[1-(4-azepan-1-yl-4-oxobutanoyl)-L-prolyl]pyrrolidine-2-carbonitrile | 50% inhibition at 0.76 nM | Sus scrofa | |
3.4.21.26 | (2R)-1-[1-(4-oxo-4-pyrrolidin-1-ylbutanoyl)-L-prolyl]pyrrolidine-2-carbonitrile | 50% inhibition at 2.9 nM | Sus scrofa | |
3.4.21.26 | (2R)-1-[1-(5-azepan-1-yl-3,3-dimethyl-5-oxopentanoyl)-L-prolyl]pyrrolidine-2-carbonitrile | 50% inhibition at 0.39 nM | Sus scrofa | |
3.4.21.26 | (2R)-1-[1-(5-azepan-1-yl-5-oxopentanoyl)-L-prolyl]pyrrolidine-2-carbonitrile | 50% inhibition at 1.2 nM | Sus scrofa |
EC Number | Organism | UniProt | Comment | Textmining |
---|---|---|---|---|
3.4.21.26 | Sus scrofa | P23687 | - |
- |
EC Number | Source Tissue | Comment | Organism | Textmining |
---|---|---|---|---|
3.4.21.26 | brain | - |
Sus scrofa | - |