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Literature summary extracted from

  • Komissarov, A.A.; Declerck, P.J.; Shore, J.D.
    Protonation State of a Single Histidine Residue Contributes Significantly to the Kinetics of the Reaction of Plasminogen Activator Inhibitor-1 with Tissue-type Plasminogen Activator (2004), J. Biol. Chem., 279, 23007-23013.
    View publication on PubMed

Inhibitors

EC Number Inhibitors Comment Organism Structure
3.4.21.68 N-((2-(iodoacetoxy)ethyl)-N-methyl)amino-7-nitrobenz-2-oxa-3-diazole P9 plasminogen activator inhibitor-1 Homo sapiens

Molecular Weight [Da]

EC Number Molecular Weight [Da] Molecular Weight Maximum [Da] Comment Organism
3.4.21.68 63500
-
x * 63500, SDS-PAGE Homo sapiens

Natural Substrates/ Products (Substrates)

EC Number Natural Substrates Organism Comment (Nat. Sub.) Natural Products Comment (Nat. Pro.) Rev. Reac.
3.4.21.68 plasminogen + H2O Homo sapiens
-
plasmin + ?
-
?

Organism

EC Number Organism UniProt Comment Textmining
3.4.21.68 Homo sapiens P00750
-
-

Source Tissue

EC Number Source Tissue Comment Organism Textmining

Substrates and Products (Substrate)

EC Number Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
3.4.21.68 plasminogen + H2O
-
Homo sapiens plasmin + ?
-
?

Subunits

EC Number Subunits Comment Organism
3.4.21.68 ? x * 63500, SDS-PAGE Homo sapiens

Synonyms

EC Number Synonyms Comment Organism
3.4.21.68 Tissue-type plasminogen activator
-
Homo sapiens
3.4.21.68 tPA
-
Homo sapiens