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Literature summary extracted from

  • Eleuteri, A.M.; Angeletti, M.; Lupidi, G.; Tacconi, R.; Bini, L.; Fioretti, E.
    Isolation and characterization of bovine thymus multicatalytic proteinase complex (2000), Protein Expr. Purif., 18, 160-168.
    View publication on PubMed

Inhibitors

EC Number Inhibitors Comment Organism Structure
3.4.25.1 3,4-dichloroisocoumarin benzyloxycarbonyl-GGL-4-nitroanilide as substrate Bos taurus
3.4.25.1 benzyloxycarbonyl-GPAF aldehyde
-
Bos taurus
3.4.25.1 benzyloxycarbonyl-GPFL aldehyde
-
Bos taurus
3.4.25.1 benzyloxycarbonyl-LLF aldehyde
-
Bos taurus

KM Value [mM]

EC Number KM Value [mM] KM Value Maximum [mM] Substrate Comment Organism Structure
3.4.25.1 0.14
-
benzyloxycarbonyl-GPALG-4-aminobenzoate enzyme from spleen Bos taurus
3.4.25.1 0.38
-
benzyloxycarbonyl-GPAFG-4-aminobenzoate enzyme from spleen Bos taurus
3.4.25.1 0.57
-
benzyloxycarbonyl-GPALG-4-aminobenzoate enzyme from thymus Bos taurus
3.4.25.1 0.8
-
benzyloxycarbonyl-GPAFG-4-aminobenzoate enzyme from thymus Bos taurus
3.4.25.1 2.29
-
benzyloxycarbonyl-GGF-4-aminobenzoate enzyme from thymus Bos taurus
3.4.25.1 3.3
-
benzyloxycarbonyl-GPAFG-4-aminobenzoate enzyme from pituitary Bos taurus

Organism

EC Number Organism UniProt Comment Textmining
3.4.25.1 Bos taurus
-
-
-

Purification (Commentary)

EC Number Purification (Comment) Organism
3.4.25.1
-
Bos taurus

Source Tissue

EC Number Source Tissue Comment Organism Textmining
3.4.25.1 thymus
-
Bos taurus
-

Substrates and Products (Substrate)

EC Number Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
3.4.25.1 benzyloxycarbonyl-D-Ala-Leu-Arg-4-nitroanilide + H2O
-
Bos taurus ?
-
?
3.4.25.1 benzyloxycarbonyl-GAPLG-p-aminobenzoate + H2O
-
Bos taurus ?
-
?
3.4.25.1 benzyloxycarbonyl-GGF-4-aminobenzoate + H2O
-
Bos taurus ?
-
?
3.4.25.1 benzyloxycarbonyl-GGF-p-aminobenzoate + H2O
-
Bos taurus ?
-
?
3.4.25.1 benzyloxycarbonyl-GGL-2-naphthylamide + H2O
-
Bos taurus ?
-
?
3.4.25.1 benzyloxycarbonyl-GPAFG-4-aminobenzoate + H2O
-
Bos taurus ?
-
?
3.4.25.1 benzyloxycarbonyl-GPAFG-p-aminobenzoate + H2O
-
Bos taurus ?
-
?
3.4.25.1 benzyloxycarbonyl-GPAGG-4-nitroanilide + H2O
-
Bos taurus ?
-
?
3.4.25.1 benzyloxycarbonyl-GPALG-4-aminobenzoate + H2O
-
Bos taurus ?
-
?
3.4.25.1 benzyloxycarbonyl-GPALG-p-aminobenzoate + H2O
-
Bos taurus ?
-
?
3.4.25.1 benzyloxycarbonyl-LLE-2-naphthylamide + H2O
-
Bos taurus ?
-
?

Turnover Number [1/s]

EC Number Turnover Number Minimum [1/s] Turnover Number Maximum [1/s] Substrate Comment Organism Structure
3.4.25.1 0.03 0.55 benzyloxycarbonyl-GPALG-4-aminobenzoate enzyme from thymus Bos taurus
3.4.25.1 0.2
-
benzyloxycarbonyl-GGF-4-aminobenzoate enzyme from thymus Bos taurus
3.4.25.1 0.5
-
benzyloxycarbonyl-GPALG-4-aminobenzoate enzyme from spleen Bos taurus
3.4.25.1 1.98
-
benzyloxycarbonyl-GPAFG-4-aminobenzoate enzyme from pituitary Bos taurus
3.4.25.1 2.94
-
benzyloxycarbonyl-GPAFG-4-aminobenzoate enzyme from pituitary Bos taurus
3.4.25.1 3
-
benzyloxycarbonyl-GPAFG-4-aminobenzoate enzyme from thymus Bos taurus
3.4.25.1 3.75
-
benzyloxycarbonyl-GPALG-4-aminobenzoate enzyme from pituitary Bos taurus
3.4.25.1 7.04
-
benzyloxycarbonyl-GPALG-4-aminobenzoate enzyme from thymus Bos taurus
3.4.25.1 12.9
-
benzyloxycarbonyl-GPALG-4-aminobenzoate enzyme from spleen Bos taurus
3.4.25.1 18.8
-
benzyloxycarbonyl-GPAFG-4-aminobenzoate enzyme from spleen Bos taurus

Ki Value [mM]

EC Number Ki Value [mM] Ki Value maximum [mM] Inhibitor Comment Organism Structure
3.4.25.1 0.00005
-
benzyloxycarbonyl-GPFL aldehyde enzyme from thymus, substrate: benzyloxycarbonyl-GPAFG-p-aminobenzoate Bos taurus
3.4.25.1 0.00082
-
benzyloxycarbonyl-GPFL aldehyde enzyme from thymus, substrate: benzyloxycarbonyl-GPALG-p-aminobenzoate Bos taurus
3.4.25.1 0.00104
-
benzyloxycarbonyl-GPFL aldehyde enzyme from spleen, substrate: benzyloxycarbonyl-GPALG-p-aminobenzoate Bos taurus
3.4.25.1 0.0016
-
benzyloxycarbonyl-LLF aldehyde enzyme from pituitary, substrate: benzyloxycarbonyl-GGF-p-aminobenzoate Bos taurus
3.4.25.1 0.002
-
benzyloxycarbonyl-GPAF aldehyde enzyme from thymus, substrate: benzyloxycarbonyl-GPALG-aminobenzoate Bos taurus
3.4.25.1 0.00251
-
benzyloxycarbonyl-LLF aldehyde enzyme from thymus, substrate: benzyloxycarbonyl-GGF-p-aminobenzoate Bos taurus
3.4.25.1 0.0026
-
benzyloxycarbonyl-GPAF aldehyde enzyme from spleen, substrate: benzyloxycarbonyl-GPALG-aminobenzoate Bos taurus
3.4.25.1 0.00466
-
benzyloxycarbonyl-GPFL aldehyde enzyme from pituitary, substrate: benzyloxycarbonyl-GPALG-p-aminobenzoate Bos taurus
3.4.25.1 0.00546
-
benzyloxycarbonyl-GPFL aldehyde enzyme from thymus, substrate: benzyloxycarbonyl-GGF-p-aminobenzoate Bos taurus
3.4.25.1 0.00597
-
benzyloxycarbonyl-LLF aldehyde enzyme from spleen, substrate: benzyloxycarbonyl-GGF-p-aminobenzoate Bos taurus
3.4.25.1 0.0162
-
benzyloxycarbonyl-GPFL aldehyde enzyme from spleen, substrate: benzyloxycarbonyl-GGF-p-aminobenzoate Bos taurus
3.4.25.1 0.0527
-
benzyloxycarbonyl-GPFL aldehyde enzyme from pituitary, substrate: benzyloxycarbonyl-GGF-p-aminobenzoate Bos taurus