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Literature summary extracted from

  • Veeraragavan, K.; Gagnon, C.
    Leupeptin and chymostatin inhibit mammalian protein methylesterase activity (1987), Biochem. Biophys. Res. Commun., 142, 603-608.
    View publication on PubMed

Inhibitors

EC Number Inhibitors Comment Organism Structure
3.1.1.61 chymostatin
-
Rattus norvegicus
3.1.1.61 D-Phe-Pro-Arg-H
-
Rattus norvegicus
3.1.1.61 leupeptin
-
Rattus norvegicus
3.1.1.61 N-tert-Butoxycarbonyl-Gln-Leu-Lys-H
-
Rattus norvegicus
3.1.1.61 pepstatin
-
Rattus norvegicus

Organism

EC Number Organism UniProt Comment Textmining
3.1.1.61 Rattus norvegicus
-
-
-

Purification (Commentary)

EC Number Purification (Comment) Organism
3.1.1.61
-
Rattus norvegicus

Source Tissue

EC Number Source Tissue Comment Organism Textmining
3.1.1.61 kidney
-
Rattus norvegicus
-

Ki Value [mM]

EC Number Ki Value [mM] Ki Value maximum [mM] Inhibitor Comment Organism Structure
3.1.1.61 0.000035
-
leupeptin pH 6.0, 37°C Rattus norvegicus
3.1.1.61 0.00054
-
chymostatin pH 6.0, 37°C Rattus norvegicus