EC Number | Inhibitors | Comment | Organism | Structure |
---|---|---|---|---|
3.4.21.75 | antipain | - |
Homo sapiens | |
3.4.21.75 | antipain | - |
Mus musculus | |
3.4.21.75 | Arg-oxime | - |
Homo sapiens | |
3.4.21.75 | Arg-oxime | - |
Mus musculus | |
3.4.21.75 | Ca2+ | 100 mM; activation below | Homo sapiens | |
3.4.21.75 | Ca2+ | 100 mM; activation below | Mus musculus | |
3.4.21.75 | CDTA | - |
Homo sapiens | |
3.4.21.75 | CDTA | - |
Mus musculus | |
3.4.21.75 | EDTA | - |
Homo sapiens | |
3.4.21.75 | EDTA | - |
Mus musculus | |
3.4.21.75 | EGTA | - |
Homo sapiens | |
3.4.21.75 | EGTA | - |
Mus musculus | |
3.4.21.75 | leupeptin | moderately | Homo sapiens | |
3.4.21.75 | leupeptin | moderately | Mus musculus | |
3.4.21.75 | Lys-Arg chloromethyl ketone | - |
Homo sapiens | |
3.4.21.75 | Lys-Arg chloromethyl ketone | - |
Mus musculus | |
3.4.21.75 | additional information | not: pepstatin | Homo sapiens | |
3.4.21.75 | additional information | not: pepstatin | Mus musculus | |
3.4.21.75 | NaCl | 600 mM | Homo sapiens | |
3.4.21.75 | NaCl | 600 mM | Mus musculus | |
3.4.21.75 | p-hydroxymercuribenzoate | - |
Homo sapiens | |
3.4.21.75 | p-hydroxymercuribenzoate | - |
Mus musculus | |
3.4.21.75 | phenylmethanesulfonyl fluoride | not | Homo sapiens | |
3.4.21.75 | phenylmethanesulfonyl fluoride | not | Mus musculus | |
3.4.21.75 | tosyl-Lys chloromethyl ketone | - |
Homo sapiens | |
3.4.21.75 | tosyl-Lys chloromethyl ketone | - |
Mus musculus |
EC Number | KM Value [mM] | KM Value Maximum [mM] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|---|
3.4.21.75 | additional information | - |
additional information | - |
Mus musculus | |
3.4.21.75 | additional information | - |
additional information | - |
Homo sapiens |
EC Number | Metals/Ions | Comment | Organism | Structure |
---|---|---|---|---|
3.4.21.75 | Ca2+ | required | Mus musculus | |
3.4.21.75 | Ca2+ | required | Homo sapiens | |
3.4.21.75 | Ca2+ | 2.46 mM | Mus musculus | |
3.4.21.75 | Ca2+ | 2.46 mM | Homo sapiens |
EC Number | Organism | UniProt | Comment | Textmining |
---|---|---|---|---|
3.4.21.75 | Homo sapiens | - |
rat somatomammotroph cell line, GH4C1 infected with vaccinia virus recombinants of human PC1 | - |
3.4.21.75 | Mus musculus | - |
rat somatomammotroph cell line, GH4C1 infected with vaccinia virus recombinants of murine PC1 | - |
EC Number | Purification (Comment) | Organism |
---|---|---|
3.4.21.75 | partial | Mus musculus |
EC Number | Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|---|
3.4.21.75 | Acetyl-Arg-Ser-Lys-Arg-4-methylcoumarin 7-amide + H2O | - |
Mus musculus | ? | - |
? | |
3.4.21.75 | Acetyl-Arg-Ser-Lys-Arg-4-methylcoumarin 7-amide + H2O | - |
Homo sapiens | ? | - |
? | |
3.4.21.75 | pGlu-Arg-Thr-Lys-Arg-4-methylcoumarin 7-amide + H2O | - |
Mus musculus | pGlu-Arg-Thr-Lys-Arg + 7-amino-4-methylcoumarin | - |
? | |
3.4.21.75 | pGlu-Arg-Thr-Lys-Arg-4-methylcoumarin 7-amide + H2O | - |
Homo sapiens | pGlu-Arg-Thr-Lys-Arg + 7-amino-4-methylcoumarin | - |
? | |
3.4.21.75 | tert-butoxycarbonyl-Arg-Val-Arg-Arg-4-methylcoumarin 7-amide + H2O | - |
Mus musculus | tert-butoxycarbonyl-Arg-Val-Arg-Arg + 7-amino-4-methylcoumarin | - |
? | |
3.4.21.75 | tert-butoxycarbonyl-Arg-Val-Arg-Arg-4-methylcoumarin 7-amide + H2O | - |
Homo sapiens | tert-butoxycarbonyl-Arg-Val-Arg-Arg + 7-amino-4-methylcoumarin | - |
? |
EC Number | Subunits | Comment | Organism |
---|---|---|---|
3.4.21.75 | ? | x * 80000-85000, mouse, SDS-PAGE | Mus musculus |
EC Number | pH Optimum Minimum | pH Optimum Maximum | Comment | Organism |
---|---|---|---|---|
3.4.21.75 | 6 | - |
acetyl-Arg-Ser-Lys-Arg-4-methylcoumaryl 7-amide | Mus musculus |
3.4.21.75 | 6 | - |
acetyl-Arg-Ser-Lys-Arg-4-methylcoumaryl 7-amide | Homo sapiens |
EC Number | pH Minimum | pH Maximum | Comment | Organism |
---|---|---|---|---|
3.4.21.75 | 5 | 6.5 | 5: about 35% of activity maximum, 6.5: about 15% of activity maximum, mouse, acetyl-Arg-Ser-Lys-Arg-4-methylcoumarin 7-amide | Mus musculus |
3.4.21.75 | 5 | 6.5 | 5: about 35% of activity maximum, 6.5: about 15% of activity maximum, mouse, acetyl-Arg-Ser-Lys-Arg-4-methylcoumarin 7-amide | Homo sapiens |