Inhibitors | Comment | Organism | Structure |
---|---|---|---|
arsenate | competitive | Mus musculus | |
GSH | competitive | Mus musculus | |
GSSG | competitive | Mus musculus | |
leukotriene D4 | competitive | Mus musculus | |
MK571 | competitive | Mus musculus | |
S-(2,4-dinitrophenyl)glutathione | competitive | Mus musculus | |
S-(p-azidophenylacyl)-glutathione | competitive | Mus musculus |
KM Value [mM] | KM Value Maximum [mM] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
0.000035 | - |
leukotriene C4/in | - |
Mus musculus | |
0.0042 | - |
vincristine/in | - |
Mus musculus | |
0.0044 | - |
etoposide/in | - |
Mus musculus | |
0.0063 | - |
daunorubicin/in | - |
Mus musculus | |
0.038 | - |
ATP | - |
Mus musculus |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Mus musculus | - |
- |
- |
Source Tissue | Comment | Organism | Textmining |
---|---|---|---|
NIH-3T3 cell | NIH 3T3 MRP transfectant pSRalpha-MRP-32 cells | Mus musculus | - |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
daunorubicin/in + ATP + H2O | - |
Mus musculus | daunorubicin/out + ADP + phosphate | - |
? | |
etoposide/in + ATP + H2O | - |
Mus musculus | etoposide/out + ADP + phosphate | - |
? | |
leukotriene C4/in + ATP + H2O | - |
Mus musculus | leukotriene C4/out + ADP + phosphate | - |
? | |
taxol/in + ATP + H2O | weak activity | Mus musculus | taxol/out + ADP + H2O | - |
? | |
vinblastine/in + ATP + H2O | weak activity | Mus musculus | vinblastine/out + ADP + phosphate | - |
? | |
vincristine/in + ATP + H2O | - |
Mus musculus | vincristine/out + ADP + phosphate | - |
? |