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Literature summary for 5.6.2.1 extracted from

  • Hackbarth, J.S.; Galvez-Peralta, M.; Dai, N.T.; Loegering, D.A.; Peterson, K.L.; Meng, X.W.; Karnitz, L.M.; Kaufmann, S.H.
    Mitotic phosphorylation stimulates DNA relaxation activity of human topoisomerase I (2008), J. Biol. Chem., 283, 16711-16722.
    View publication on PubMedView publication on EuropePMC

Protein Variants

Protein Variants Comment Organism
S10A/S112A/S394A triple mutant 3A Homo sapiens
S10A/S21A/S112A/S394A quadruple phosphomutant 4A Homo sapiens
S21A site-directed mutagenesis Homo sapiens
Y723F site-directed mutagenesis Homo sapiens

Inhibitors

Inhibitors Comment Organism Structure
camptothecin
-
Homo sapiens

Organism

Organism UniProt Comment Textmining
Homo sapiens
-
-
-

Source Tissue

Source Tissue Comment Organism Textmining
A-549 cell human lung cancer cells Homo sapiens
-
K-562 cell human leukemia cells Homo sapiens
-

Synonyms

Synonyms Comment Organism
topoI
-
Homo sapiens
Topoisomerase I
-
Homo sapiens