Any feedback?
Please rate this page
(literature.php)
(0/150)

BRENDA support

Literature summary for 5.6.2.1 extracted from

  • Riou, G.; Douc-Rasy, S.; Kayser, A.
    Inhibitors of trypanosome topoisomerases (1986), Biochem. Soc. Trans., 14, 496-499.
    View publication on PubMed

Inhibitors

Inhibitors Comment Organism Structure
9-Hydroxyellipticine
-
Trypanosoma cruzi
9-Hydroxyellipticine
-
Trypanosoma equiperdum
Acriflavine
-
Trypanosoma cruzi
Acriflavine
-
Trypanosoma equiperdum
Berenil
-
Trypanosoma cruzi
Berenil
-
Trypanosoma equiperdum
Clorobiocin
-
Trypanosoma cruzi
Clorobiocin
-
Trypanosoma equiperdum
coumermycin coumermycin A2 Trypanosoma cruzi
coumermycin coumermycin A2 Trypanosoma equiperdum
ellipticine
-
Trypanosoma cruzi
ellipticine
-
Trypanosoma equiperdum
Hydroxystilbamidine
-
Trypanosoma cruzi
Hydroxystilbamidine
-
Trypanosoma equiperdum
Lampit
-
Trypanosoma cruzi
Lampit
-
Trypanosoma equiperdum

Organism

Organism UniProt Comment Textmining
Trypanosoma cruzi
-
-
-
Trypanosoma equiperdum
-
-
-

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
supercoiled DNA relaxation Trypanosoma cruzi relaxed closed circular DNA
-
?
supercoiled DNA relaxation Trypanosoma equiperdum relaxed closed circular DNA
-
?