Inhibitors | Comment | Organism | Structure |
---|---|---|---|
rofecoxib | inhibitor of cyclooxygenase COX-2, additionally non-competitive inhibition of prostacyclin synthase in aortic microsomal fractions. No significant inhibition up to 0.001 mM | Bos taurus | |
rofecoxib | inhibitor of cyclooxygenase COX-2, additionally non-competitive inhibition of prostacyclin synthase | Homo sapiens |
Localization | Comment | Organism | GeneOntology No. | Textmining |
---|---|---|---|---|
microsome | - |
Bos taurus | - |
- |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Bos taurus | - |
- |
- |
Homo sapiens | - |
- |
- |
Source Tissue | Comment | Organism | Textmining |
---|---|---|---|
aorta | - |
Bos taurus | - |
HUVEC cell | - |
Homo sapiens | - |
umbilical vein endothelial cell | - |
Homo sapiens | - |
IC50 Value | IC50 Value Maximum | Comment | Organism | Inhibitor | Structure |
---|---|---|---|---|---|
0.001 | - |
22°C, 0.001 mM rofecoxib completely blocks cyclooxygenase COX-2 | Homo sapiens | rofecoxib | |
0.01 | - |
22°C. No significant inhibition up to 0.001 mM | Bos taurus | rofecoxib |