Literature summary for 5.2.1.8 extracted from

Andres, C.J.; Macdonald, T.L.
Conformationally defined analogs of prolylamides. trans-Prolyl peptidomimetics (1993), J. Org. Chem., 58, 6609-6613.

No PubMed abstract available

Inhibitors

Inhibitors	Comment	Organism	Structure
(E)-2-(2-hydroxy-2-isobutylethy 1idene)-1-meth ylcyclopentane-(L)-tyrosylcarboxamide	-	Homo sapiens

Organism	UniProt	Comment	Textmining
Homo sapiens	-	isoform FKBP12, recombinant protein	-

Ki Value [mM]	Ki Value maximum [mM]	Inhibitor	Comment	Organism	Structure
0.0086	-	(E)-2-(2-hydroxy-2-isobutylethy 1idene)-1-meth ylcyclopentane-(L)-tyrosylcarboxamide	0°C, pH 8.0	Homo sapiens

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Release 2023.1 (January 2023)