Inhibitors | Comment | Organism | Structure |
---|---|---|---|
additional information | amphotericin B, fluconazole, ketoconazole or allopurinol do not significantly affect ATPase and/or ADPase activity of promastigotes preparation, no or poor to low (at high concentrations) inhibition | Leishmania infantum | |
pentamidine isethionate | PEN, inhibits 74% and 35% of the ATPase and ADPase activities, respectively of the purified enzyme NTPDase 1, no inhibition of NTPDase 2 | Leishmania infantum |
Metals/Ions | Comment | Organism | Structure |
---|---|---|---|
Ca2+ | activates | Leishmania infantum |
Natural Substrates | Organism | Comment (Nat. Sub.) | Natural Products | Comment (Nat. Pro.) | Rev. | Reac. |
---|---|---|---|---|---|---|
ADP + H2O | Leishmania infantum | - |
AMP + phosphate | - |
? | |
ADP + H2O | Leishmania infantum MHOM/BR/1972/BH46 | - |
AMP + phosphate | - |
? | |
ATP + H2O | Leishmania infantum | - |
ADP + phosphate | - |
? | |
ATP + H2O | Leishmania infantum MHOM/BR/1972/BH46 | - |
ADP + phosphate | - |
? |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Leishmania infantum | - |
- |
- |
Leishmania infantum MHOM/BR/1972/BH46 | - |
- |
- |
Source Tissue | Comment | Organism | Textmining |
---|---|---|---|
amastigote | - |
Leishmania infantum | - |
additional information | propagated in macrophages | Leishmania infantum | - |
promastigote | - |
Leishmania infantum | - |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
ADP + H2O | - |
Leishmania infantum | AMP + phosphate | - |
? | |
ADP + H2O | - |
Leishmania infantum MHOM/BR/1972/BH46 | AMP + phosphate | - |
? | |
ATP + H2O | - |
Leishmania infantum | ADP + phosphate | - |
? | |
ATP + H2O | - |
Leishmania infantum MHOM/BR/1972/BH46 | ADP + phosphate | - |
? |
Synonyms | Comment | Organism |
---|---|---|
NTPDase 1 | - |
Leishmania infantum |
nucleoside triphosphate diphosphohydrolase 1 | - |
Leishmania infantum |
Temperature Optimum [°C] | Temperature Optimum Maximum [°C] | Comment | Organism |
---|---|---|---|
37 | - |
assay at | Leishmania infantum |
pH Optimum Minimum | pH Optimum Maximum | Comment | Organism |
---|---|---|---|
7.4 | - |
assay at | Leishmania infantum |